NCT01319773

Brief Summary

This study will evaluate the safety, tolerability and pharmacokinetics of two formulations of cyclosporine ophthalmic emulsion in healthy adults (parallel-group phase). The parallel-group phase will be followed by a paired-eye phase which will evaluate the safety and tolerability of two formulations of cyclosporine ophthalmic emulsion compared with cyclosporine ophthalmic emulsion (RESTASIS®) in patients with dry eye.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
44

participants targeted

Target at P50-P75 for phase_1

Timeline
Completed

Started Nov 2010

Shorter than P25 for phase_1

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

November 1, 2010

Completed
2 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 1, 2011

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

January 1, 2011

Completed
3 months until next milestone

First Submitted

Initial submission to the registry

March 18, 2011

Completed
4 days until next milestone

First Posted

Study publicly available on registry

March 22, 2011

Completed
12 months until next milestone

Results Posted

Study results publicly available

March 2, 2012

Completed
Last Updated

September 7, 2015

Status Verified

August 1, 2015

Enrollment Period

2 months

First QC Date

March 18, 2011

Results QC Date

January 31, 2012

Last Update Submit

August 25, 2015

Conditions

Outcome Measures

Primary Outcomes (1)

  • Concentration of Cyclosporine Measured in Blood at Day 1 in the Parallel-Group Phase (PGP)

    Concentration of cyclosporine measured in blood at Day 1 of the parallel-group phase (PGP). Blood samples were collected up to 3 hours post-dose and concentrations of cyclosporine were measured.

    Day 1

Secondary Outcomes (2)

  • Number of Subjects Who Reported Ocular Symptoms During the Parallel-Group Phase (PGP)

    3 Days

  • Number of Eyes With Ocular Symptoms Post-Dose During the Paired-Eye Phase (PEP) at Day 1

    Day 1

Study Arms (5)

cyclosporine ophthalmic emulsion Formulation A (Formulation A)

EXPERIMENTAL

Parallel-Group Phase (PGP): cyclosporine ophthalmic emulsion Formulation A

Drug: cyclosporine ophthalmic emulsion Formulation A

cyclosporine ophthalmic emulsion Formulation B (Formulation B)

EXPERIMENTAL

PGP: cyclosporine ophthalmic emulsion Formulation B

Drug: cyclosporine ophthalmic emulsion Formulation B

Formulation A and cyclosporine ophthalmic emulsion 0.05%

OTHER

Paired-Eye Phase (PEP): cyclosporine ophthalmic emulsion Formulation A and cyclosporine ophthalmic emulsion 0.05%

Drug: cyclosporine ophthalmic emulsion Formulation A; cyclosporine ophthalmic emulsion 0.05%

Formulation B and cyclosporine ophthalmic emulsion 0.05%

OTHER

PEP: cyclosporine ophthalmic emulsion Formulation B and cyclosporine ophthalmic emulsion 0.05%

Drug: cyclosporine ophthalmic emulsion Formulation B; cyclosporine ophthalmic emulsion 0.05%

Formulation A and Formulation B

EXPERIMENTAL

PEP: cyclosporine ophthalmic emulsion Formulation A and cyclosporine ophthalmic emulsion Formulation B

Drug: cyclosporine ophthalmic emulsion Formulation A; cyclosporine ophthalmic emulsion Formulation B

Interventions

One drop of cyclosporine ophthalmic emulsion Formulation A administered to each eye twice daily for 2 days and once in the morning of Day 3.

cyclosporine ophthalmic emulsion Formulation A (Formulation A)

One drop of cyclosporine ophthalmic emulsion Formulation B administered to each eye twice daily for 2 days and once in the morning of Day 3.

cyclosporine ophthalmic emulsion Formulation B (Formulation B)

One drop of cyclosporine ophthalmic emulsion Formulation A administered to one eye and one drop of cyclosporine ophthalmic emulsion 0.05% administered to the opposite eye, twice daily for 1 day.

Also known as: RESTASIS®
Formulation A and cyclosporine ophthalmic emulsion 0.05%

One drop of cyclosporine ophthalmic emulsion Formulation B administered to one eye and one drop of cyclosporine ophthalmic emulsion 0.05% administered to the opposite eye, twice daily for 1 day.

Also known as: RESTASIS®
Formulation B and cyclosporine ophthalmic emulsion 0.05%

One drop of cyclosporine ophthalmic emulsion Formulation A administered to one eye and one drop of cyclosporine ophthalmic emulsion Formulation B administered to the opposite eye, twice daily for 1 day.

Formulation A and Formulation B

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Parallel-Group Phase:
  • Weigh at least 110 lbs
  • to 45 years old
  • Paired-Eye Phase:
  • Dry eye disease in both eyes

You may not qualify if:

  • Parallel-Group Phase:
  • Use of nicotine products, any medications, supplements or herbal products or consumption of grapefruit juice within 14 days or anticipated use during the study
  • Has donated blood within 90 days
  • Significant weight change (over 10 lbs) within 60 days
  • Previous use of RESTASIS®
  • Parallel-Group and Paired-Eye Phases:
  • Anticipated wearing of contact lenses during the study or wearing of contact lenses within 14 days
  • Consumption of alcohol products within 72 hours
  • Paired-Eye Phase:
  • Previous ocular surgery
  • Use of RESTASIS® within 30 days

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Unknown Facility

Newport Beach, California, United States

Location

MeSH Terms

Conditions

Dry Eye Syndromes

Interventions

Cyclosporins

Condition Hierarchy (Ancestors)

Lacrimal Apparatus DiseasesEye Diseases

Intervention Hierarchy (Ancestors)

Peptides, CyclicMacrocyclic CompoundsPolycyclic CompoundsPeptidesAmino Acids, Peptides, and Proteins

Results Point of Contact

Title
Therapeutic Area Head
Organization
Allergan, Inc.

Study Officials

  • Medical Director

    Allergan

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, INVESTIGATOR, OUTCOMES ASSESSOR
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 18, 2011

First Posted

March 22, 2011

Study Start

November 1, 2010

Primary Completion

January 1, 2011

Study Completion

January 1, 2011

Last Updated

September 7, 2015

Results First Posted

March 2, 2012

Record last verified: 2015-08

Locations