NCT01281462

Brief Summary

This is a study in adult subjects with complicated urinary tract infection (cUTI) comparing treatment with intravenous (IV) coadministered ceftaroline fosamil and NXL104 versus treatment with IV doripenem.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
217

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Dec 2010

Geographic Reach
7 countries

50 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

December 1, 2010

Completed
1 month until next milestone

First Submitted

Initial submission to the registry

January 13, 2011

Completed
11 days until next milestone

First Posted

Study publicly available on registry

January 24, 2011

Completed
1.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 1, 2012

Completed
4 months until next milestone

Study Completion

Last participant's last visit for all outcomes

July 1, 2012

Completed
Last Updated

February 3, 2014

Status Verified

January 1, 2014

Enrollment Period

1.2 years

First QC Date

January 13, 2011

Last Update Submit

January 2, 2014

Conditions

Keywords

complicated Urinary Tract InfectionAcute Pyelonephritis

Outcome Measures

Primary Outcomes (2)

  • Microbiological response of Microbiologically Evaluable (ME) at Test of Cure (TOC)

    The number and percentage of subjects in each treatment group recorded as having a favorable microbiological response in the ME Population at Test-of-Cure (TOC)

    5 to 11 days after last dose of study drug

  • Evaluate safety

    Evaluate the safety of coadministered IV ceftaroline fosamil and NXL104 in subjects with cUTI. Summaries of AEs, SAEs, deaths, laboratory evaluations (hematology and coagulation studies, comprehensive metabolic panel, and urinalysis), vital signs, ECGs, and physical examinations will be provided for each treatment group.

    from administration of first dose of study drug to the Late -Follow -Up (LFU) visit (28 to 42 days after administration of the last dose of study drug)

Secondary Outcomes (1)

  • Clinical response in CE at Test of Cure

    5 to 11 days after last dose of study drug

Study Arms (3)

Ceftaroline fosamil and NXL104 (q8h)

EXPERIMENTAL
Drug: Ceftaroline fosamil and NXL104 (q8h)Drug: Placebo

Ceftaroline fosamil and NXL104 (q12h)

EXPERIMENTAL
Drug: Ceftaroline fosamil and NXL104 (q12h)Drug: Placebo

Doripenem

ACTIVE COMPARATOR
Drug: DoripenemDrug: Placebo

Interventions

600 mg ceftaroline fosamil/600 mg NXL104 IV coadministered every 8 hours (q8h);

Also known as: Ceftaroline fosamil and Avibactam(NXL104) (q8h)
Ceftaroline fosamil and NXL104 (q8h)

600 mg ceftaroline fosamil/600 mg NXL104 IV coadministered every 12 hours (q12h);

Also known as: Ceftaroline fosamil and Avibactam(NXL104) (q12h)
Ceftaroline fosamil and NXL104 (q12h)

500 mg doripenem IV q8h;

Doripenem

On CXL-MD-02, there were (3) treatment arms (meaning a subject could be randomized to 1 of 3 possible treatment regimens). Each treatment arm contained 1 or 2 placebo doses of IV saline in order to preserve the blind.

Also known as: placebo (saline)
Ceftaroline fosamil and NXL104 (q12h)Ceftaroline fosamil and NXL104 (q8h)Doripenem

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Have pyuria (white blood cells in the urine)
  • Clinical signs and/or symptoms of cUTI (including acute pyelonephritis)
  • Have a pretreatment baseline urine culture specimen
  • The subject's infection would require initial treatment with IV antibiotics
  • The subject must require initial hospitalization to manage the cUTI by the standard of care.

You may not qualify if:

  • History of any hypersensitivity or allergic reaction to any β-lactam (eg, cephalosporins, penicillins, carbapenems)
  • Confirmed fungal urinary tract infection
  • Intractable UTI anticipated to require more than 10 days of study drug therapy
  • Complete, permanent obstruction of the urinary tract\\
  • Permanent indwelling bladder catheter or instrumentation (including nephrostomy) or current urinary catheter that will not be removed during IV study drug administration
  • Suspected or confirmed perinephric or intrarenal abscess
  • Suspected or confirmed prostatitis
  • Ileal loops or vesico-ureteral reflux
  • Impairment of renal function including a calculated CrCl of \< 30 mL/min, requirement for peritoneal dialysis, hemodialysis or hemofiltration, or oliguria
  • Renal transplantation
  • Life expectancy less than 3 months
  • Evidence of significant hepatic, hematological, or immunologic disease or dysfunction
  • Past or current history of epilepsy or seizure disorder
  • Women who are pregnant or nursing

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (50)

Investigational Site

La Mesa, California, 91942, United States

Location

Investigational Site

San Diego, California, 92120, United States

Location

Investigational Site

Pensacola, Florida, 32504, United States

Location

Investigational Site

Baltimore, Maryland, 21287, United States

Location

Investigational Site

Detroit, Michigan, 48202, United States

Location

Investigational Site

Plovdiv, 4002, Bulgaria

Location

Investigational Site

Rousse, 7002, Bulgaria

Location

Investigational Site

Sofia, 1407, Bulgaria

Location

Investigational Site

Sofia, 1431, Bulgaria

Location

Investigational Site

Sofia, 1606, Bulgaria

Location

Investigational Site

Varna, 9002, Bulgaria

Location

Investigational Site

Berlin, 10117, Germany

Location

Investigational Site

Freiburg im Breisgau, 79106, Germany

Location

Investigational Site

Giessen, 35385, Germany

Location

Investigational Site

Kassel, 34125, Germany

Location

Investigational Site

Minden, 32429, Germany

Location

Investigational Site

Müllheim, 79379, Germany

Location

Investigational Site

Paderborn, 33098, Germany

Location

Investigational Site

Planegg, 82152, Germany

Location

Investigational Site

Beirut, Lebanon

Location

Investigational Site

Bialystok, 15-950, Poland

Location

Investigational Site

Bielsko-Biala, 43-316, Poland

Location

Investigational Site

Częstochowa, 42-200, Poland

Location

Investigational Site

Katowice, 40-073, Poland

Location

Investigational Site

Katowice, 40-752, Poland

Location

Investigational Site

Lodz, 90-153, Poland

Location

Investigational Site

Tychy, 43-100, Poland

Location

Investigational Site

Warsaw, 03-401, Poland

Location

Investigational Site

Wołomin, 05-200, Poland

Location

Investigational Site

Wroclaw, 50-349, Poland

Location

Investigational Site

Zamość, 22-400, Poland

Location

Investigational Site

Moscow, 105077, Russia

Location

Investigational Site

Moscow, 105425, Russia

Location

Investigational Site

Moscow, 111123, Russia

Location

Investigational Site

Moscow, 119049, Russia

Location

Investigational Site

Moscow, 119992-119435, Russia

Location

Investigational Site

Rostov-on-Don, 344022, Russia

Location

Investigational Site

Saint Petersburg, 193312, Russia

Location

Investigational Site

Saint Petersburg, 194044, Russia

Location

Investigational Site

Saint Petersburg, 194291, Russia

Location

Investigational Site

Saint Petersburg, 194354, Russia

Location

Investigational Site

Saint Petersburg, 195067, Russia

Location

Investigational Site

Saint Petersburg, 196247, Russia

Location

Investigational Site

Saint Petersburg, 198205, Russia

Location

Investigational Site

Saint Petersburg, 199178, Russia

Location

Investigational Site

Smolensk, 214018, Russia

Location

Investigational Site

Diyarbakır, 21280, Turkey (Türkiye)

Location

Investigational Site

Eskişehir, 26480, Turkey (Türkiye)

Location

Investigational Site

Izmir, 35040, Turkey (Türkiye)

Location

Investigational Site

Izmir, 35340, Turkey (Türkiye)

Location

MeSH Terms

Conditions

Urinary Tract Infections

Interventions

CeftarolineavibactamDoripenemSodium Chloride

Condition Hierarchy (Ancestors)

InfectionsUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital Diseases

Intervention Hierarchy (Ancestors)

Cephalosporinsbeta-LactamsLactamsAmidesOrganic ChemicalsThiazinesSulfur CompoundsHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingHeterocyclic CompoundsCarbapenemsChloridesHydrochloric AcidChlorine CompoundsInorganic ChemicalsSodium Compounds

Study Officials

  • Medical Monitor

    Forest Laboratories

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 13, 2011

First Posted

January 24, 2011

Study Start

December 1, 2010

Primary Completion

March 1, 2012

Study Completion

July 1, 2012

Last Updated

February 3, 2014

Record last verified: 2014-01

Locations