NCT01251848

Brief Summary

The study is to assess if sitaxsentan and ritonavir will affect the blood levels of each other when coadministered.

Trial Health

15
At Risk

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Trial has exceeded expected completion date
Timeline
Completed

Started Jan 2011

Shorter than P25 for phase_1

Status
withdrawn

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

December 1, 2010

Completed
1 day until next milestone

First Posted

Study publicly available on registry

December 2, 2010

Completed
1 month until next milestone

Study Start

First participant enrolled

January 1, 2011

Completed
1 month until next milestone

Primary Completion

Last participant's last visit for primary outcome

February 1, 2011

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

February 1, 2011

Completed
Last Updated

March 5, 2015

Status Verified

March 1, 2015

Enrollment Period

1 month

First QC Date

December 1, 2010

Last Update Submit

March 4, 2015

Conditions

Keywords

Sitaxentanritonavirdrug interactionpharmacokinetics

Outcome Measures

Primary Outcomes (4)

  • The comparison of peak plasma concentration of sitaxsentan when coadministered with ritonavir versus sitaxsentan administered alone.

    24 hours

  • The comparison of area under the curve of sitaxsentan when coadministered with ritonavir versus sitaxsentan administered alone.

    24 hours

  • The comparison of peak plasma concentration of ritonavir when coadministered with sitaxsentan versus ritonavir administered alone.

    24 hours

  • The comparison of area under the curve of ritonavir when coadministered with sitaxsentan versus ritonavir administered alone.

    24 hours

Study Arms (3)

Treatment A

ACTIVE COMPARATOR
Drug: Sitaxentan

Treatment B

ACTIVE COMPARATOR
Drug: Ritonavir

Treatment C

EXPERIMENTAL
Drug: SitaxsentanDrug: Ritonavir

Interventions

Sitaxsentan Tablet, 100 mg, q24h (once daily) for 5 days.

Treatment A

Ritonavir Capsule, 100 mg, q12h (twice daily) for 5 days (morning dose only on Day 5).

Treatment B

Sitaxsentan Tablet, 100 mg, q24h (once daily) for 5 days

Treatment C

Eligibility Criteria

Age21 Years - 55 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Healthy male subjects and/or women of non-child bearing potential.
  • Subjects (because of teratogenic risk of sitaxsentan) between the ages of 21 and 55 years, inclusive.
  • Signed informed consent.

You may not qualify if:

  • Evidence or history of clinically significant hematological, renal, endocrine, pulmonary, gastrointestinal, cardiovascular, hepatic, psychiatric, neurologic, or allergic disease.
  • History of significant alcohol and drug use.
  • Has hepatic dysfunction.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Related Links

MeSH Terms

Conditions

Pulmonary Arterial Hypertension

Interventions

sitaxsentanRitonavir

Condition Hierarchy (Ancestors)

Hypertension, PulmonaryLung DiseasesRespiratory Tract Diseases

Intervention Hierarchy (Ancestors)

ThiazolesSulfur CompoundsOrganic ChemicalsAzolesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR
0

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
NONE
Purpose
BASIC SCIENCE
Intervention Model
CROSSOVER
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

December 1, 2010

First Posted

December 2, 2010

Study Start

January 1, 2011

Primary Completion

February 1, 2011

Study Completion

February 1, 2011

Last Updated

March 5, 2015

Record last verified: 2015-03