NCT01096667

Brief Summary

MK-8835-042 (B1521004) is designed to assess the safety and efficacy of an investigational drug, ertugliflozin (MK-8835, PF-04971729), in participants with type 2 diabetes and hypertension. Participants in the study will receive 1 of 5 treatments for 28 days (either placebo, 1 of 3 doses of ertugliflozin \[1, 5, or 25 mg\], or the approved drug hydrochlorothiazide \[HCTZ\]). The primary hypothesis of the study was that ertugliflozin was superior to placebo on the change from baseline in average, 24-hour systolic blood pressure (SBP) on Day 28.

Trial Health

100
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
194

participants targeted

Target at P50-P75 for phase_2 diabetes-mellitus-type-2

Timeline
Completed

Started May 2010

Shorter than P25 for phase_2 diabetes-mellitus-type-2

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

March 26, 2010

Completed
5 days until next milestone

First Posted

Study publicly available on registry

March 31, 2010

Completed
2 months until next milestone

Study Start

First participant enrolled

May 17, 2010

Completed
9 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

February 9, 2011

Completed
16 days until next milestone

Study Completion

Last participant's last visit for all outcomes

February 25, 2011

Completed
6.8 years until next milestone

Results Posted

Study results publicly available

December 13, 2017

Completed
Last Updated

September 13, 2018

Status Verified

August 1, 2018

Enrollment Period

9 months

First QC Date

March 26, 2010

Results QC Date

November 15, 2017

Last Update Submit

August 15, 2018

Conditions

Keywords

type 2 diabeteshypertensionambulatory blood pressure monitoring

Outcome Measures

Primary Outcomes (2)

  • Baseline 24-hour Average Systolic Blood Pressure (SBP)

    Baseline 24-hour average SBP was assessed using 24-hour ambulatory blood pressure monitoring (ABPM).

    24 hours

  • Change From Baseline on 24-hour Average SBP at Week 4

    Change from baseline on 24-hour average SBP at Week 4 assessed using 24-hour ABPM. In the case of missing data, last observation carried forward (LOCF).

    Baseline and Week 4

Secondary Outcomes (24)

  • Baseline Average Daytime and Nighttime SBP

    Daytime: 16 hours; Nighttime: 8 hours

  • Change From Baseline on Daytime Average SBP at Week 4

    Baseline and Week 4

  • Change From Baseline on Nighttime Average SBP at Week 4

    Baseline and Week 4

  • Baseline Seated, Triplicate Trough SBP

    Baseline

  • Change From Baseline in Seated, Triplicate Trough SBP at Week 4

    Baseline and Week 4

  • +19 more secondary outcomes

Study Arms (5)

Placebo

PLACEBO COMPARATOR

Placebo to ertugliflozin (resembling either 1 mg or 5 mg), placebo to ertugliflozin (resembling 25 mg), and placebo to HCTZ once daily for 28 days.

Drug: Placebo to Ertuglilflozin 1 or 5 mgDrug: Placebo to HCTZDrug: Placebo to ertuglilflozin 25 mg

Ertugliflozin 1 mg

EXPERIMENTAL

Ertugliflozin 1 mg, placebo to ertugliflozin (resembling 25 mg), and placebo to HCTZ once daily for 28 days

Drug: Ertugliflozin 1 mgDrug: Placebo to HCTZDrug: Placebo to ertuglilflozin 25 mg

Ertugliflozin 5 mg

EXPERIMENTAL

Ertugliflozin 5 mg, placebo to ertugliflozin (resembling 25 mg), and placebo to HCTZ once daily for 28 days

Drug: Ertugliflozin 5 mgDrug: Placebo to HCTZDrug: Placebo to ertuglilflozin 25 mg

Ertugliflozin 25 mg

EXPERIMENTAL

Ertugliflozin 25 mg, placebo to ertugliflozin (resembling either 1 mg or 5 mg), and placebo to HCTZ once daily for 28 days

Drug: Placebo to Ertuglilflozin 1 or 5 mgDrug: Ertugliflozin 25 mgDrug: Placebo to HCTZ

HCTZ 12.5mg

ACTIVE COMPARATOR

HCTZ 12.5 mg, placebo to ertugliflozin (resembling either 1 mg or 5 mg), and placebo to ertugliflozin (resembling 25 mg) once daily for 28 days

Drug: Placebo to Ertuglilflozin 1 or 5 mgDrug: HCTZ 12.5mgDrug: Placebo to ertuglilflozin 25 mg

Interventions

Placebo to ertuglilflozin tablet 1 or 5 mg once daily for 28 days

Ertugliflozin 25 mgHCTZ 12.5mgPlacebo

Ertugliflozin tablet 1 mg once daily for 28 days

Ertugliflozin 1 mg

Ertugliflozin tablet 5 mg once daily for 28 days

Ertugliflozin 5 mg

Ertugliflozin tablet 25 mg once daily for 28 days

Ertugliflozin 25 mg

Hydrocholorthiazide (HCTZ) 12.5 mg capsule once daily for 28 days

HCTZ 12.5mg

Placebo to HCTZ 12.5 mg capsule once daily for 28 days

Ertugliflozin 1 mgErtugliflozin 25 mgErtugliflozin 5 mgPlacebo

Placebo to ertuglilflozin tablet 25 mg once daily for 28 days

Ertugliflozin 1 mgErtugliflozin 5 mgHCTZ 12.5mgPlacebo

Eligibility Criteria

Age18 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Participants with type 2 diabetes and hypertension
  • Medically stable
  • On at least 1 (and up to 2) oral diabetes drugs
  • And up to 2 medicines for blood pressure control

You may not qualify if:

  • Participants with type 1 diabetes
  • Heart attack
  • Stroke
  • Uncontrolled blood pressure
  • Significant kidney disease

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Related Publications (2)

  • Amin NB, Wang X, Mitchell JR, Lee DS, Nucci G, Rusnak JM. Blood pressure-lowering effect of the sodium glucose co-transporter-2 inhibitor ertugliflozin, assessed via ambulatory blood pressure monitoring in patients with type 2 diabetes and hypertension. Diabetes Obes Metab. 2015 Aug;17(8):805-8. doi: 10.1111/dom.12486. Epub 2015 Jun 17.

  • Fediuk DJ, Sahasrabudhe V, Dawra VK, Zhou S, Sweeney K. Population Pharmacokinetic Analyses of Ertugliflozin in Select Ethnic Populations. Clin Pharmacol Drug Dev. 2021 Nov;10(11):1297-1306. doi: 10.1002/cpdd.970. Epub 2021 Jul 2.

MeSH Terms

Conditions

Diabetes Mellitus, Type 2Hypertension

Interventions

ertugliflozinHydrochlorothiazide

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System DiseasesVascular DiseasesCardiovascular Diseases

Intervention Hierarchy (Ancestors)

ChlorothiazideBenzothiadiazinesSulfonamidesSulfonesSulfur CompoundsOrganic ChemicalsThiazidesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingHeterocyclic Compounds

Results Point of Contact

Title
Senior Vice President, Global Clinical Development
Organization
Merck Sharp & Dohme Corp.

Study Officials

  • Medical Director

    Merck Sharp & Dohme LLC

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 26, 2010

First Posted

March 31, 2010

Study Start

May 17, 2010

Primary Completion

February 9, 2011

Study Completion

February 25, 2011

Last Updated

September 13, 2018

Results First Posted

December 13, 2017

Record last verified: 2018-08

Data Sharing

IPD Sharing
Will share

https://www.merck.com/clinical-trials/pdf/ProcedureAccessClinicalTrialData.pdf

More information