NCT00952445

Brief Summary

The purpose of the study is to determine if repeated daily doses of T0903131 (INT131) Besylate over 4 weeks can lower fasting blood glucose in patients with Type 2 Diabetes Mellitus.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
70

participants targeted

Target at P50-P75 for phase_2

Timeline
Completed

Started Dec 2003

Shorter than P25 for phase_2

Geographic Reach
1 country

21 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

December 1, 2003

Completed
6 months until next milestone

Study Completion

Last participant's last visit for all outcomes

June 1, 2004

Completed
5.2 years until next milestone

First Submitted

Initial submission to the registry

August 4, 2009

Completed
2 days until next milestone

First Posted

Study publicly available on registry

August 6, 2009

Completed
Last Updated

October 19, 2022

Status Verified

October 1, 2022

First QC Date

August 4, 2009

Last Update Submit

October 17, 2022

Conditions

Study Arms (3)

T0903131 Besylate

EXPERIMENTAL

1.0 mg

Drug: T0903131 Besylate

T0903131 Besylate (higher dose)

EXPERIMENTAL

10.0 mg

Drug: T0903131 Besylate

Placebo

PLACEBO COMPARATOR

Once daily, oral

Drug: Placebo

Interventions

Once daily, oral

Placebo

Once daily, oral

Also known as: INT131 Besylate
T0903131 BesylateT0903131 Besylate (higher dose)

Eligibility Criteria

Age30 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Clinical Diagnosis of Type 2 Diabetes Mellitus for at least 3 months prior to enrollment
  • Fasting Plasma Glucose between 126 and 240 mg/dL
  • Hemoglobin-A1c (HbA1c) between 6.8% and 10.0%
  • Fasting C-peptide \> 0.8 ng/mL

You may not qualify if:

  • Treatment with any pharmacotherapy for Type 2 Diabetes Mellitus within previous 6 weeks prior to screening
  • Prior treatment with Thiazolidinedione, including Troglitazone, Rosiglitazone, pioglitazone
  • BMI \> 42 kg/m2
  • Presence of any diabetic complications requiring chronic therapy
  • Presence or history of any form of hepatic disease
  • Serum creatinine \> 1.8 mg/dL
  • History of cardiac arrhythmias or abnormal cardiac electrophysiology
  • Any reason that, in the Investigator's judgment, would have interfered with the ability of the subject to comply with the requirements of the protocol

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (21)

Whittier Diabetes Institute

La Jolla, California, United States

Location

Charles R. Drew University

Los Angeles, California, United States

Location

National Research Institute

Los Angeles, California, United States

Location

Lovelace Research Institute

Santa Ana, California, United States

Location

University of Miami

Miami, Florida, United States

Location

GFI Research Center

Evansville, Indiana, United States

Location

Joslin Diabetes Center

Boston, Massachusetts, United States

Location

Radiant Research

Edina, Minnesota, United States

Location

Radiant Research

St Louis, Missouri, United States

Location

St Louis Center for Clinical Research

St Louis, Missouri, United States

Location

Kaleida Health Diabetes Center

Buffalo, New York, United States

Location

Rochester Clinical Research

Rochester, New York, United States

Location

Duke University Medical Center

Durham, North Carolina, United States

Location

Radiant Research

Portland, Oregon, United States

Location

Radiant Research

Anderson, South Carolina, United States

Location

Baylor University Endocrine Center

Dallas, Texas, United States

Location

Dallas Diabetes and Endocrine Research Center

Dallas, Texas, United States

Location

Endocrine Associates of Dallas

Dallas, Texas, United States

Location

Diabetes and Grandular Disease Clinic and Reseach Center

San Antonio, Texas, United States

Location

Endocrine Research Specialists

Ogden, Utah, United States

Location

Salem VA Medical Center

Salem, Virginia, United States

Location

Related Publications (1)

  • Dunn FL, Higgins LS, Fredrickson J, DePaoli AM; INT131-004 study group. Selective modulation of PPARgamma activity can lower plasma glucose without typical thiazolidinedione side-effects in patients with Type 2 diabetes. J Diabetes Complications. 2011 May-Jun;25(3):151-8. doi: 10.1016/j.jdiacomp.2010.06.006. Epub 2010 Aug 23.

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

August 4, 2009

First Posted

August 6, 2009

Study Start

December 1, 2003

Study Completion

June 1, 2004

Last Updated

October 19, 2022

Record last verified: 2022-10

Locations