NCT00929708

Brief Summary

The purpose of this study is to investigate the efficacy, safety and tolerability of 4 weeks treatment with AZD3199 in moderate to severe COPD.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
329

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Jun 2009

Shorter than P25 for phase_2

Geographic Reach
5 countries

38 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

June 1, 2009

Completed
25 days until next milestone

First Submitted

Initial submission to the registry

June 26, 2009

Completed
3 days until next milestone

First Posted

Study publicly available on registry

June 29, 2009

Completed
8 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 1, 2010

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

March 1, 2010

Completed
3.9 years until next milestone

Results Posted

Study results publicly available

January 17, 2014

Completed
Last Updated

February 17, 2014

Status Verified

January 1, 2014

Enrollment Period

9 months

First QC Date

June 26, 2009

Results QC Date

December 20, 2012

Last Update Submit

January 22, 2014

Conditions

Keywords

COPDEfficacySafetyInhalation

Outcome Measures

Primary Outcomes (2)

  • FEV1, E0-4; the Average Value at Visit 5 From Before to 4 Hours After Morning Dose (Peak Effect)

    change from baseline

    0,5 min, 15 min, 60 min, 2 h, 4 h

  • FEV1, E24-26; the Average Value at Visit 5 Between 24 and 26 Hours Following the Morning Dose (Trough Effect)

    change from baseline

    24h, 26h

Secondary Outcomes (7)

  • Cmax; the Highest Plasma Concentration of AZD3199 Measured

    0,15 min, 1, 4 and 24 hours post dose

  • AUC0-24; Area Under the Plasma Concentration Curve From Zero to 24 Hours After Dose

    0,15 min, 1, 4 and 24 hours post dose

  • FEV1 Post Salbutamol Inhalation

    Baseline (visit 2) and 26 h after the last morning dose (visit 5).

  • Total Number of Reliever Medication Inhalations Per 24h

    During day (from rising from bed until going to bed) and night (from going to bed until rising from bed) at visit 1 to visit 5 (24h), up to 4 weeks.

  • Total AstraZeneca COPD Symptoms Scores (Included Breathlessness, Chest Tightness, Cough and Night-time Awakenings)

    Daily, during run-in and treatment

  • +2 more secondary outcomes

Study Arms (5)

1

EXPERIMENTAL

AZD3199 low dose

Drug: AZD3199

2

EXPERIMENTAL

AZD3199 intermediate dose

Drug: AZD3199

3

EXPERIMENTAL

AZD3199 high dose

Drug: AZD3199

4

ACTIVE COMPARATOR

Formoterol 2x4.5 microgram bid

Drug: formoterol

5

PLACEBO COMPARATOR

Placebo

Drug: Placebo

Interventions

Dry powder for inhalation, o.d., 4 weeks

123

Dry powder for inhalation, b.i.d., 4 weeks

4

Dry powder for inhalation, b.i.d., 4 weeks

5

Eligibility Criteria

Age40 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • COPD
  • Current or exsmokers, 10 pack years

You may not qualify if:

  • Asthma
  • Any clinically relevant abnormal findings at screening examinations
  • Recent COPD exacerbation

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (38)

Research Site

Blagoevgrad, Bulgaria

Location

Research Site

Pleven, Bulgaria

Location

Research Site

Rousse, Bulgaria

Location

Research Site

Sofia, Bulgaria

Location

Research Site

Varna, Bulgaria

Location

Research Site

Moncton, New Brunswick, Canada

Location

Research Site

St. John's, Newfoundland and Labrador, Canada

Location

Research Site

Truro, Nova Scotia, Canada

Location

Research Site

Greater Sudbury, Ontario, Canada

Location

Research Site

Mississauga, Ontario, Canada

Location

Research Site

Toronto, Ontario, Canada

Location

Research Site

Pointe-Claire, Quebec, Canada

Location

Research Site

Saint Romuald, Quebec, Canada

Location

Research Site

Trois-Rivières, Quebec, Canada

Location

Research Site

Yanagawa, Fukuoka, Japan

Location

Research Site

Fukuyama, Hiroshima, Japan

Location

Research Site

Chitose, Hokkaido, Japan

Location

Research Site

Obihiro, Hokkaido, Japan

Location

Research Site

Tomakomai, Hokkaido, Japan

Location

Research Site

Hitachi, Ibaragi, Japan

Location

Research Site

Naka-gun, Ibaraki, Japan

Location

Research Site

Sendai, Miyagi, Japan

Location

Research Site

Osaka, Osaka, Japan

Location

Research Site

Toyonaka, Osaka, Japan

Location

Research Site

Moriyama, Shiga, Japan

Location

Research Site

Ōtsu, Shiga, Japan

Location

Research Site

Machida, Tokyo, Japan

Location

Research Site

Kitakyushu, Japan

Location

Research Site

Bialystok, Poland

Location

Research Site

Gorzow Wlkp, Poland

Location

Research Site

Lodz, Poland

Location

Research Site

Lublin, Poland

Location

Research Site

Poznan, Poland

Location

Research Site

Szczecin, Poland

Location

Research Site

Tarnów, Poland

Location

Research Site

Moscow, Russia

Location

Research Site

Novosibirsk, Russia

Location

Research Site

Saint Petersburg, Russia

Location

Related Publications (1)

  • Kuna P, Ivanov Y, Trofimov VI, Saito T, Beckman O, Bengtsson T, Jorup C, Maltais F. Efficacy and safety of AZD3199 vs formoterol in COPD: a randomized, double-blind study. Respir Res. 2013 Jun 3;14(1):64. doi: 10.1186/1465-9921-14-64.

MeSH Terms

Conditions

Pulmonary Disease, Chronic ObstructiveRespiratory Aspiration

Interventions

AZD-3199Formoterol Fumarate

Condition Hierarchy (Ancestors)

Lung Diseases, ObstructiveLung DiseasesRespiratory Tract DiseasesChronic DiseaseDisease AttributesPathologic ProcessesPathological Conditions, Signs and SymptomsRespiration Disorders

Intervention Hierarchy (Ancestors)

EthanolaminesAmino AlcoholsAlcoholsOrganic ChemicalsAmines

Results Point of Contact

Title
Carin Jorup, MSD
Organization
AstraZeneca

Study Officials

  • Piotr Kuna, Professor

    University Hospital, Lodz, Poland

    PRINCIPAL INVESTIGATOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 26, 2009

First Posted

June 29, 2009

Study Start

June 1, 2009

Primary Completion

March 1, 2010

Study Completion

March 1, 2010

Last Updated

February 17, 2014

Results First Posted

January 17, 2014

Record last verified: 2014-01

Locations