NCT00746837

Brief Summary

The purpose of the study is to estimate the absolute bioavailability at steady state of 2 doses of AZD5672 (50 mg and 150 mg administered orally once daily)

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
26

participants targeted

Target at P25-P50 for phase_1 healthy-volunteers

Timeline
Completed

Started Aug 2008

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

August 1, 2008

Completed
1 month until next milestone

First Submitted

Initial submission to the registry

September 3, 2008

Completed
1 day until next milestone

First Posted

Study publicly available on registry

September 4, 2008

Completed
4 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 1, 2009

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

January 1, 2009

Completed
Last Updated

December 2, 2010

Status Verified

November 1, 2010

Enrollment Period

5 months

First QC Date

September 3, 2008

Last Update Submit

November 30, 2010

Conditions

Keywords

AZD5672

Outcome Measures

Primary Outcomes (1)

  • PK variables

    Frequent sampling occasions during study periods

Secondary Outcomes (1)

  • Safety variables (adverse events, blood pressure, pulse, safety lab)

    During the whole treatment periods

Study Arms (2)

1

EXPERIMENTAL

Single ascending IV dose, 3 treatment periods separated by a minimum 14 day washout between doses

Drug: AZD5672

2

EXPERIMENTAL

2 cohorts single IV dose + multiple oral dose period separated by a minimum of 14 days washout between IV and oral dose

Drug: AZD5672

Interventions

single IV doses starting at 7 mg, subsequent doses to be confirmed following review of PK and safety data after each treatment period

12

Eligibility Criteria

Age18 Years - 55 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Provision of informed consent prior to any study specific procedures.
  • Females should not be of childbearing potential
  • Clinically normal physical and laboratory findings as judged by the investigator, including negative test results for drug-of-abuse, alcohol and cotinine at the Screening Visit and/or admission (Day -1) of each study period, and negative test results

You may not qualify if:

  • Any clinically significant disease or disorder which, in the opinion of the investigator, may either put the subject at risk because of participation in the study, or may influence the results of the study, or the subject's ability to participate
  • Unsuitable venous access for intravenous studies
  • Participation in a clinical study involving an investigational product within 5 half-lives of active moieties of the last dose of investigational product or 3 months prior to first dosing (whichever is longer).

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Research Site

Harrow, London, United Kingdom

Location

MeSH Terms

Interventions

N-(1-(3-(3,5-difluorophenyl)-3-(4-methanesulfonylphenyl)propyl)piperidin-4-yl)-N-ethyl-2-(4-methanesulfonylphenyl)acetamide

Study Officials

  • Mark Layton, MD, PhD

    AstraZeneca R&D, Charnwood, UK

    STUDY DIRECTOR
  • Tania Hugo

    PAREXEL Clinical Pharmacology Research Unit

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
BASIC SCIENCE
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

September 3, 2008

First Posted

September 4, 2008

Study Start

August 1, 2008

Primary Completion

January 1, 2009

Study Completion

January 1, 2009

Last Updated

December 2, 2010

Record last verified: 2010-11

Locations