NCT00734032

Brief Summary

The primary objective of this study is to examine the effects of SB-480848 on plasma lipoprotein associated phospholipase A2 (Lp-PLA2) activity in dyslipidemic patients during a 4-week treatment with SB-480848.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
107

participants targeted

Target at P50-P75 for phase_2

Timeline
Completed

Started Aug 2008

Shorter than P25 for phase_2

Geographic Reach
1 country

7 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

August 12, 2008

Completed
1 day until next milestone

First Posted

Study publicly available on registry

August 13, 2008

Completed
13 days until next milestone

Study Start

First participant enrolled

August 26, 2008

Completed
5 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 16, 2009

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

January 16, 2009

Completed
9 years until next milestone

Results Posted

Study results publicly available

January 12, 2018

Completed
Last Updated

January 12, 2018

Status Verified

January 1, 2018

Enrollment Period

5 months

First QC Date

August 12, 2008

Results QC Date

July 18, 2017

Last Update Submit

January 10, 2018

Conditions

Keywords

SB-480848Dyslipidaemia

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline to Week 4 in Plasma Lipoprotein-associated Phospholipase A2 (Lp-PLA2) Activity

    Blood sample for Lp-PLA2 activity was collected before administration of study medication on the sampling day. Participants were instructed to visit without meal and study medication in the morning. The study medication was administered with food following test. Baseline value was defined as the assessment done on Week 0 (Visit 2). Change from Baseline was calculated as the post-Baseline (Week 4) assessment value minus the Baseline assessment value. If either value was missing, then the change from Baseline was set to be missing. The natural logarithm (log) was used for transformation in Lp-PLA2 activity. In case of zero values, an offset of 0.0001 was added to the zero values to ensure that the log transformation was successfully applied. The log transformation was conducted on the original value and then taken the change from Baseline on that log original value, calculated as log (post-Baseline value \[week 4\]) minus log (Baseline value).

    Baseline (Week 0, Visit 2) and Week 4

Secondary Outcomes (2)

  • Percent Inhibition of Lp-PLA2 Activity in Plasma Over Time

    Baseline (Week 0, Visit 2) up to Follow-up (up to Week 7)

  • Change From Baseline in Lp-PLA2 Activity at Week 1, 2 and Follow-up

    Baseline (Week 0, Visit 2), Week 1, Week 2 and Follow-up ( Week 7)

Study Arms (4)

Placebo Group

PLACEBO COMPARATOR

Matched Placebo

Drug: SB480848 Placebo Tablet

SB480848 40mg Group

EXPERIMENTAL

SB480848 40mg/day

Drug: SB480848 40mg EC Tablet

SB480848 80mg Group

EXPERIMENTAL

SB480848 80mg/day

Drug: SB480848 80mg EC Tablet

SB480848 160mg Group

EXPERIMENTAL

SB480848 160mg/day

Drug: SB480848 160mg EC Tablet

Interventions

1 tablet once a day

Also known as: Darapladib
SB480848 40mg Group

1 tablet once a day

SB480848 80mg Group

1 tablet once a day

SB480848 160mg Group

1 tablet once a day

Placebo Group

Eligibility Criteria

Age20 Years - 80 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Dyslipidemic subject who is currently undergoing statin therapy and no change in lipid-lowering therapy or dose during the 4 week prior to randomization

You may not qualify if:

  • Recent (i.e.,\<6 months prior to screening) CV event and/or vascular procedure defined as:
  • A)ST-elevation MI or non-ST-elevation MI B)Unstable angina C)Coronary revascularization \[(percutaneous coronary intervention (PCI) or coronary artery bypass graft (CABG)\] D)Stroke of any etiology E)Peripheral arterial disease with critical limb ischemia (resting pain or ischemic skin lesions, either ulcers or gangrene) F)Resuscitated cardiac arrest
  • Planned CABG or planned PCI or planned major non-cardiac surgery within study period
  • No measurable Lp-PLA2 activity in plasma (\<10 nmol/min/mL) at screening
  • Change in a lipid-lowering medication, regimen or dosage during the 4 week prior to randomization
  • Poorly controlled dyslipidemia (LDL-c \>=160 mg/dL) at screening

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (7)

GSK Investigational Site

Fukuoka, 812-0025, Japan

Location

GSK Investigational Site

Fukuoka, 818-0036, Japan

Location

GSK Investigational Site

Fukuoka, 819-1102, Japan

Location

GSK Investigational Site

Tokyo, 105-0004, Japan

Location

GSK Investigational Site

Tokyo, 154-0024, Japan

Location

GSK Investigational Site

Tokyo, 160-0017, Japan

Location

GSK Investigational Site

Tokyo, 174-0051, Japan

Location

Related Links

MeSH Terms

Conditions

AtherosclerosisDyslipidemias

Interventions

darapladib

Condition Hierarchy (Ancestors)

ArteriosclerosisArterial Occlusive DiseasesVascular DiseasesCardiovascular DiseasesLipid Metabolism DisordersMetabolic DiseasesNutritional and Metabolic Diseases

Results Point of Contact

Title
GSK Response Center
Organization
GlaxoSmithKline

Study Officials

  • GSK Clinical Trials

    GlaxoSmithKline

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

August 12, 2008

First Posted

August 13, 2008

Study Start

August 26, 2008

Primary Completion

January 16, 2009

Study Completion

January 16, 2009

Last Updated

January 12, 2018

Results First Posted

January 12, 2018

Record last verified: 2018-01

Data Sharing

IPD Sharing
Will share

Patient-level data for this study will be made available through www.clinicalstudydatarequest.com following the timelines and process described on this site.

Available IPD Datasets

Informed Consent Form (LPL110118)Access
Annotated Case Report Form (LPL110118)Access
Clinical Study Report (LPL110118)Access
Dataset Specification (LPL110118)Access
Individual Participant Data Set (LPL110118)Access
Statistical Analysis Plan (LPL110118)Access

Locations