NCT00686179

Brief Summary

The purpose of this study is to evaluate the effects on cardiac repolarisation of supratherapeutic doses of AZD3480 compared to placebo in healthy male volunteers, subgrouped as extensive metabolisers and poor metabolisers according to CYP2D6 metabolic capacity, using moxifloxacin as positive control.

Trial Health

100
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
75

participants targeted

Target at P75+ for phase_1 healthy

Timeline
Completed

Started Jan 2008

Typical duration for phase_1 healthy

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

January 1, 2008

Completed
5 months until next milestone

First Submitted

Initial submission to the registry

May 27, 2008

Completed
2 days until next milestone

First Posted

Study publicly available on registry

May 29, 2008

Completed
2 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 1, 2008

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

August 1, 2008

Completed
Last Updated

September 25, 2008

Status Verified

September 1, 2008

Enrollment Period

7 months

First QC Date

May 27, 2008

Last Update Submit

September 24, 2008

Conditions

Keywords

TQTECGQTQTcAZD3480ECG(QTc effects)

Outcome Measures

Primary Outcomes (1)

  • QTcX interval (supratherapeutic doses in comparison to placebo).Subject-specific correction of QT, QTcF and QTcB (supportive outcome variables).Bazett QTcB=QT*RR-1/2Fridericia QTcF=QT'RR-1/3

    11 dECG measurements x 4 (4-way crossover)

Secondary Outcomes (3)

  • QTcX (therapeutic doses in comparison to placebo).PR-, QRS-, RR-intervals

    11 dECG measurements x 4 (4-way crossover)

  • Plasma concentration (AUC, Cmax, tmax etc)

    11 PK-measurements x 4 (4-way crossover)

  • Registration of AEs, blood pressure, ECG, clinical laboratory tests

    From enrolment to follow-up

Study Arms (4)

1

EXPERIMENTAL

Escalating doses of AZD3480 during 6 days

Drug: AZD3480

2

EXPERIMENTAL

Repeated doses of AZD3480 during 6 days

Drug: AZD3480

3

PLACEBO COMPARATOR

Placebo during 6 days

Drug: PLACEBO

4

ACTIVE COMPARATOR

Placebo during 5 days, active day 6

Drug: Moxifloxacin

Interventions

Capsule, oral, single dose, 6 days

Also known as: TC-1734-226
12

Capsule(encapsulated), oral, single dose

4

Capsule, oral, single dose

3

Eligibility Criteria

Age20 Years - 60 Years
Sexmale
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Participation in a previous study for genotyping for identification to be extensive or poor metaboliser (CYP2D6 enzyme)
  • Physically and mentally healthy male volunteers

You may not qualify if:

  • History of clinically significant diseases or illness.
  • Participation in another study the last 3 months
  • Prescribed or non-prescribed medications from 3 weeks prior to first treatment day until follow-up except for paracetamol (max 1.5 g per day.)

Contact the study team to confirm eligibility.

Sponsors & Collaborators

MeSH Terms

Interventions

isproniclineMoxifloxacin

Intervention Hierarchy (Ancestors)

Fluoroquinolones4-QuinolonesQuinolonesQuinolinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingHeterocyclic Compounds

Study Officials

  • Hans-Göran Hårdemark

    Clinical Neuroscience TA AstraZeneca R&D Södertälje, Sweden

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
PREVENTION
Intervention Model
CROSSOVER
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

May 27, 2008

First Posted

May 29, 2008

Study Start

January 1, 2008

Primary Completion

August 1, 2008

Study Completion

August 1, 2008

Last Updated

September 25, 2008

Record last verified: 2008-09