NCT00684190

Brief Summary

The purpose of the study is to evaluate if AZD3355 and Nexium interact with each other or not, i.e. show the same or altered plasma concentration profiles when co-administered compared to administered alone.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
30

participants targeted

Target at P25-P50 for phase_1

Timeline
Completed

Started Mar 2008

Shorter than P25 for phase_1

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

March 1, 2008

Completed
3 months until next milestone

First Submitted

Initial submission to the registry

May 22, 2008

Completed
4 days until next milestone

First Posted

Study publicly available on registry

May 26, 2008

Completed
6 days until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 1, 2008

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

June 1, 2008

Completed
Last Updated

December 3, 2010

Status Verified

December 1, 2010

Enrollment Period

3 months

First QC Date

May 22, 2008

Last Update Submit

December 2, 2010

Conditions

Keywords

Reflux InhibitorGERDPPI Interaction

Outcome Measures

Primary Outcomes (1)

  • PK variables

    Frequent sampling occasions during day 7 each treatment period

Secondary Outcomes (2)

  • 4-BOH cholesterol

    Sampling occasions during day 7 one treatment period (AZD3355 alone)

  • Safety variables (adverse events, blood pressure, pulse, safety lab)

    During the whole treatment period

Study Arms (3)

1

EXPERIMENTAL

AZD3355 150 mg

Drug: AZD3355

2

EXPERIMENTAL

Esomeprazole 40mg

Drug: Esomeprazole

3

EXPERIMENTAL

AZD3355 150mg/Esomeprazole 40mg

Drug: AZD3355Drug: Esomeprazole

Interventions

150 mg bid, oral, 7 days

Also known as: Lesogaberan
13

40 mg od, oral, 7 days

Also known as: Nexium
23

Eligibility Criteria

Age18 Years - 45 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Provision of written informed consent
  • Females no childbearing potential
  • Clinically normal physical findings

You may not qualify if:

  • Clinically significant illness within 2 weeks prior to the first dose of investigational product
  • History of clinically significant disease
  • Use of prescribed medication during the 2 weeks before administration of the first dose of investigational product

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Research Site

Uppsala, Sweden

Location

Related Publications (1)

  • Niazi M, Silberg DG, Miller F, Ruth M, Holmberg AA. Evaluation of the pharmacokinetic interaction between lesogaberan (AZD3355) and esomeprazole in healthy subjects. Drugs R D. 2010;10(4):243-51. doi: 10.2165/11588180-000000000-00000.

MeSH Terms

Conditions

Gastroesophageal Reflux

Interventions

lesogaberanEsomeprazole

Condition Hierarchy (Ancestors)

Esophageal Motility DisordersDeglutition DisordersEsophageal DiseasesGastrointestinal DiseasesDigestive System Diseases

Intervention Hierarchy (Ancestors)

Omeprazole2-PyridinylmethylsulfinylbenzimidazolesSulfoxidesSulfur CompoundsOrganic ChemicalsPyridinesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsBenzimidazolesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-Ring

Study Officials

  • Eva Ersdal, PhD

    AstraZeneca R&D, Mölndal, Sweden

    STUDY DIRECTOR
  • Jan Vouis, MD

    Quintiles AB, Uppsala, Sweden

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
NONE
Purpose
BASIC SCIENCE
Intervention Model
CROSSOVER
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

May 22, 2008

First Posted

May 26, 2008

Study Start

March 1, 2008

Primary Completion

June 1, 2008

Study Completion

June 1, 2008

Last Updated

December 3, 2010

Record last verified: 2010-12

Locations