NCT00678145

Brief Summary

Intensive glucose control in type 1 diabetes mellitus (T1DM) is associated with clear health benefits (1). However, despite development of insulin analogs, pump/multi-dose treatment and continuous glucose monitoring, maintaining near-normal glycemia remains an elusive goal for most patients, in large part owing to the risk of hypoglycemia. T1DM patients are susceptible to hypoglycemia due to defective counterregulatory responses (CR) characterized by: 1) deficient glucagon release during impending/early hypoglycemia; 2) additional hypoglycemia-associated autonomic failure (HAAF) and exercise-associated autonomic failure (EAAF) that blunt the sympathoadrenal responses to hypoglycemia following repeated episodes of hypoglycemia or exercise as well as degrading other CR; and 3) hypoglycemia unawareness (HU), lowering the threshold for symptoms that trigger behavioral responses (e.g. eating). Thus, the risk of hypoglycemia in T1DM impedes ideal insulin treatment and leads to defaulting to suboptimal glycemic control (2). There are two approaches that could resolve this important clinical problem: 1) perfection of glucose sensing and insulin and glucagon delivery approaches (bioengineered or cell-based) that mimic normal islet function and precisely regulate glucose continuously, or 2) a drug to enhance or normalize the pattern of CR to hypoglycemia. Despite much research and important advances in the field, neither islet transplantation nor biosensor devices have emerged as viable long-term solutions for the majority of patients (3, 4). Over the past several years, our lab has explored the approach of enhancing CR by examining mechanisms responsible for HAAF/EAAF and searching for potential pharmacological methods to modulate the CR to hypoglycemia (5-11). Our work has led to a paradigm shift in the field of hypoglycemia, exemplified by the novel hypothesis and published experimental data supporting a role for opioid signaling that resulted in the initiation of exploratory clinical trials by other research groups.

Trial Health

43
At Risk

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Trial has exceeded expected completion date
Enrollment
116

participants targeted

Target at P50-P75 for phase_2 diabetes-mellitus

Timeline
Completed

Started Mar 2008

Longer than P75 for phase_2 diabetes-mellitus

Geographic Reach
1 country

1 active site

Status
unknown

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

March 1, 2008

Completed
2 months until next milestone

First Submitted

Initial submission to the registry

May 14, 2008

Completed
1 day until next milestone

First Posted

Study publicly available on registry

May 15, 2008

Completed
14.2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 1, 2022

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

August 1, 2022

Completed
Last Updated

January 14, 2021

Status Verified

January 1, 2021

Enrollment Period

14.4 years

First QC Date

May 14, 2008

Last Update Submit

January 12, 2021

Conditions

Keywords

DiabetesHypoglycemiaHAAFCounterregulation

Outcome Measures

Primary Outcomes (1)

  • Change in the counterregulatory responses to hypoglycemia compared to controls

    Measurements of counterregulatory hormones will be measured throughout the study

    Measured every 15 minutes at timepoints 0, 15, 30, 45...120 through study completion

Secondary Outcomes (1)

  • Symptom scores

    Measured every 15 minutes at timepoints 0, 15, 30, 45...120 through study completion

Study Arms (2)

Healthy

EXPERIMENTAL

Healthy individuals will receive drug (naloxone, morphine sulfate, epinephrine) and placebo comparator.

Drug: naloxoneDietary Supplement: fructoseBehavioral: exerciseDrug: Morphine sulfateDrug: Epinephrine

Type 1 Diabetes

EXPERIMENTAL

T1D individuals will receive drug (naloxone, morphine sulfate, epinephrine) and placebo comparator.

Drug: naloxoneDietary Supplement: fructoseBehavioral: exerciseDrug: Morphine sulfateDrug: Epinephrine

Interventions

Administering naloxone on Day 1, and quantifying the counterregulatory responses to hypoglycemia on Day 2.

Also known as: Narcan
HealthyType 1 Diabetes
fructoseDIETARY_SUPPLEMENT

Administering fructose on Day 1, and quantifying the counterregulatory responses to hypoglycemia on Day 2.

Also known as: Insulin
HealthyType 1 Diabetes
exerciseBEHAVIORAL

Administering exercise on Day 1, and quantifying the counterregulatory responses to hypoglycemia on Day 2.

HealthyType 1 Diabetes

Administering morphine on Day 1, and quantifying the counterregulatory responses to hypoglycemia on Day 2.

Also known as: Morphine
HealthyType 1 Diabetes

Administering epinephrine on Day 1, and quantifying the counterregulatory responses to hypoglycemia on Day 2.

Also known as: Adrenalin
HealthyType 1 Diabetes

Eligibility Criteria

Age21 Years - 60 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Non-diabetic individuals

You may not qualify if:

  • Hypertension
  • Hyperlipidemia
  • Heart disease
  • Cerebrovascular disease
  • Seizures
  • Bleeding disorders

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Albert Einstein College of Medicine / General Clinical Research Center

The Bronx, New York, 10461, United States

Location

Related Publications (2)

  • Carey M, Gospin R, Goyal A, Tomuta N, Sandu O, Mbanya A, Lontchi-Yimagou E, Hulkower R, Shamoon H, Gabriely I, Hawkins M. Opioid Receptor Activation Impairs Hypoglycemic Counterregulation in Humans. Diabetes. 2017 Nov;66(11):2764-2773. doi: 10.2337/db16-1478. Epub 2017 Aug 31.

  • Milman S, Leu J, Shamoon H, Vele S, Gabriely I. Opioid receptor blockade prevents exercise-associated autonomic failure in humans. Diabetes. 2012 Jun;61(6):1609-15. doi: 10.2337/db11-1622. Epub 2012 Apr 20.

MeSH Terms

Conditions

Diabetes MellitusHypoglycemiaPure Autonomic Failure

Interventions

NaloxoneFructoseInsulinExerciseMorphineEpinephrine

Condition Hierarchy (Ancestors)

Glucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System DiseasesPrimary DysautonomiasAutonomic Nervous System DiseasesNervous System Diseases

Intervention Hierarchy (Ancestors)

MorphinansOpiate AlkaloidsAlkaloidsHeterocyclic CompoundsHeterocyclic Compounds, Bridged-RingHeterocyclic Compounds, 4 or More RingsHeterocyclic Compounds, Fused-RingPhenanthrenesPolycyclic Aromatic HydrocarbonsPolycyclic CompoundsHexosesMonosaccharidesSugarsCarbohydratesKetosesProinsulinInsulinsPancreatic HormonesPeptide HormonesHormonesHormones, Hormone Substitutes, and Hormone AntagonistsPeptidesAmino Acids, Peptides, and ProteinsMotor ActivityMovementMusculoskeletal Physiological PhenomenaMusculoskeletal and Neural Physiological PhenomenaMorphine DerivativesEthanolaminesAmino AlcoholsAlcoholsOrganic ChemicalsAminesBiogenic MonoaminesBiogenic AminesCatecholaminesCatecholsPhenolsBenzene DerivativesHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbons

Study Officials

  • Meredith Hawkins, M.D., M.S.

    Albert Einstein College of Medicine

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
BASIC SCIENCE
Intervention Model
CROSSOVER
Sponsor Type
OTHER
Responsible Party
PRINCIPAL INVESTIGATOR
PI Title
Principal Investigator

Study Record Dates

First Submitted

May 14, 2008

First Posted

May 15, 2008

Study Start

March 1, 2008

Primary Completion

August 1, 2022

Study Completion

August 1, 2022

Last Updated

January 14, 2021

Record last verified: 2021-01

Data Sharing

IPD Sharing
Will not share

Locations