NCT00559871

Brief Summary

The purpose of this study is to determine whether Fipamezole is effective in the treatment of levodopa-induced dyskinesia in advanced Parkinson's disease.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
180

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Oct 2007

Geographic Reach
2 countries

36 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

October 1, 2007

Completed
2 months until next milestone

First Submitted

Initial submission to the registry

November 15, 2007

Completed
1 day until next milestone

First Posted

Study publicly available on registry

November 16, 2007

Completed
1.5 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 1, 2009

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

May 1, 2009

Completed
Last Updated

June 3, 2009

Status Verified

June 1, 2009

Enrollment Period

1.6 years

First QC Date

November 15, 2007

Last Update Submit

June 2, 2009

Conditions

Keywords

dyskinesiamovement disordersbasal ganglia diseasesJP-1730Parkinsonend-of-dose wearing offfluctuations

Outcome Measures

Primary Outcomes (1)

  • To compare the efficacy of 3 different doses of fipamezole with that of placebo on dyskinesia as assessed by a dyskinesia assessment scale.

    28-days treatment

Secondary Outcomes (1)

  • To compare efficacy of 3 different doses of fipamezole with that of placebo on the mean daily 'Off' time, as recorded in the patient diary.

    28-days treatment

Study Arms (4)

1

PLACEBO COMPARATOR

One placebo tablet administered tid from Day 1 to 28

Drug: fipamezole

2

ACTIVE COMPARATOR

One 30-mg tablet of Fipamezole tid from Day 1 to 28

Drug: fipamezole

3

ACTIVE COMPARATOR

One 30-mg tablet of Fipamezole tid from Day 1 to 7; and one 60-mg tablet of Fipamezole tid from Day 8 to 28

Drug: fipamezole

4

ACTIVE COMPARATOR

One 30-mg tablet of Fipamezole tid from Day 1 to 7; one 60-mg tablet of Fipamezole tid from Day 8 to 14; and one 90-mg tablet of Fipamezole tid from Day 15 to 28

Drug: fipamezole

Interventions

Fipamezole in Zydis formulation three times per day for up to 28 days

Also known as: JP-1730
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Eligibility Criteria

Age30 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Idiopathic Parkinson's disease.
  • Levodopa/DDI associated peak-dose dyskinesia which is at least moderately disabling and present for ≥25% of the waking day (UPDRS part IV, items 32 and 33, each ≥ 2).
  • Stable Parkinson's medication for at least 1 month prior to randomization.
  • Hoehn and Yahr Stages 1 to 4 during 'Off' period.
  • Demonstrated ability to comprehend and give informed consent.
  • Ability to complete patient diary.

You may not qualify if:

  • Other clinically significant conditions apart from those typically associated with Parkinson's disease.
  • Intake of medication associated with exacerbation of dyskinesia or with extrapyramidal side effects and tardive dyskinesia or induction of liver enzymes; neuroleptics; or specified drugs known to be substantially metabolized through the following cytochrome P450 isoenzymes: 1A2, 2B6, 2C19, 2C9, 2D6, and 2E1.
  • Use of St. John's Wort or Ginkgo Biloba within 48 hrs prior to randomization and until the last treatment day with the study medication.
  • Intake of an investigational drug within 30 days prior to initial screening.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (36)

University of Alabama at Birmingham

Birmingham, Alabama, 35233, United States

Location

Neurology Clinic PC

Northport, Alabama, 35476, United States

Location

University of Arizona Health Sciences Center

Tucson, Arizona, 85724-5023, United States

Location

Parkinson and Movement Disorder Institute

Fountain Valley, California, 92708, United States

Location

University of California Irvine

Irvine, California, 92697, United States

Location

Coastal Neurological Medicine Group

La Jolla, California, 92037, United States

Location

Colorado Neurological Institute

Englewood, Colorado, 80113, United States

Location

Parkinson's Disease and Movement Disorder Center

Boca Raton, Florida, 33486, United States

Location

Sunrise Clinical Research

Hollywood, Florida, 33021, United States

Location

Pharmax Research Clinic

Miami, Florida, 33126, United States

Location

University of Miami

Miami, Florida, 33136, United States

Location

Collier Neurological Clinic

Naples, Florida, 34102, United States

Location

University of South Florida, Parkinson's Disease and Movement Center

Tampa, Florida, 33606, United States

Location

Emory Healthcare

Atlanta, Georgia, 30329, United States

Location

Medical College of Georgia

Augusta, Georgia, 30912, United States

Location

Rush University Medical Center

Chicago, Illinois, 60612, United States

Location

Parkinson Disease Center - University of Kansas Medical Center

Kansas City, Kansas, 66160, United States

Location

Ochsner Clinic Foundation

New Orleans, Louisiana, 70121, United States

Location

Maryland Parkinson's Disease and Movement Disorder Center

Baltimore, Maryland, 21201, United States

Location

U Mass Memorial Medical Center

Worcester, Massachusetts, 01655-0318, United States

Location

Henry Ford Health Systems, Franklin Pointe Medical Center

Southfield, Michigan, 48034, United States

Location

Struthers Parkinson's Center

Golden Valley, Minnesota, 55427, United States

Location

Neurology Group of Bergen County

Ridgewood, New Jersey, 07450, United States

Location

Biomedical Research Alliance of New York

Forest Hills, New York, 11375, United States

Location

Duke Health Center at Morreene Road

Durham, North Carolina, 27705, United States

Location

Oregon Health and Science University

Portland, Oregon, 97239-3098, United States

Location

Semmes Murphey Neurologic and Spine Institute

Memphis, Tennessee, 38104, United States

Location

Baylor College of Medicine

Houston, Texas, 77030, United States

Location

Neurology Associates

San Antonio, Texas, 78258, United States

Location

Max Superspecialty Hospital

Saket, New Delhi, 110017, India

Location

Neurology centre

Ahmedabad, 380006, India

Location

St John's Medical College & Hospital

Bangalore, 560 034, India

Location

M S Ramaiah Medical College Hospital

Bangalore, 560 054, India

Location

Nizam's Institute of Medical Sciences

Hyderabaad, 500 082, India

Location

Chatrapati Sahuji Maharaj Medical University

Lucknow, 226003, India

Location

J.S.S. Medical College and Hospital

Mysore, 570 004, India

Location

MeSH Terms

Conditions

Parkinson DiseaseDyskinesiasMovement DisordersBasal Ganglia Diseases

Interventions

fipamezole

Condition Hierarchy (Ancestors)

Parkinsonian DisordersBrain DiseasesCentral Nervous System DiseasesNervous System DiseasesSynucleinopathiesNeurodegenerative DiseasesNeurologic ManifestationsSigns and SymptomsPathological Conditions, Signs and Symptoms

Study Officials

  • Peter A. LeWitt, M.D.

    Henry Ford Health Systems, Franklin Pointe Medical Center

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

November 15, 2007

First Posted

November 16, 2007

Study Start

October 1, 2007

Primary Completion

May 1, 2009

Study Completion

May 1, 2009

Last Updated

June 3, 2009

Record last verified: 2009-06

Locations