NCT00492232

Brief Summary

The purpose of this study is to assess whether ramelteon, once daily (QD), can facilitate the discontinuation of zolpidem in subjects with chronic insomnia.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
135

participants targeted

Target at P50-P75 for phase_4

Timeline
Completed

Started Apr 2007

Shorter than P25 for phase_4

Geographic Reach
1 country

41 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

April 1, 2007

Completed
3 months until next milestone

First Submitted

Initial submission to the registry

June 25, 2007

Completed
2 days until next milestone

First Posted

Study publicly available on registry

June 27, 2007

Completed
8 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 1, 2008

Completed
2 months until next milestone

Study Completion

Last participant's last visit for all outcomes

May 1, 2008

Completed
1.2 years until next milestone

Results Posted

Study results publicly available

July 17, 2009

Completed
Last Updated

July 20, 2010

Status Verified

July 1, 2010

Enrollment Period

11 months

First QC Date

June 25, 2007

Results QC Date

May 28, 2009

Last Update Submit

July 13, 2010

Conditions

Keywords

Chronic InsomniaSleep Initiation and Maintenance DisorderDrug Therapy

Outcome Measures

Primary Outcomes (1)

  • Percentage of Participants Who Discontinued Zolpidem Therapy

    Participants reduced zolpidem incrementally from Week 3 to Week 10 of the double-blind treatment period (DBTP). A participant who did not take any zolpidem during the last 7 days of the DBTP was defined as having completely discontinued zolpidem by that time point. The number of subjects who discontinued zolpidem at the end of the DBTP was summarized.

    Week 10

Secondary Outcomes (13)

  • Change From Baseline in Weekly Zolpidem Dosage During Weeks 1-2

    Baseline and Weeks 1-2

  • Change From Baseline in Weekly Zolpidem Dosage During Weeks 3-4

    Baseline and Weeks 3-4

  • Change From Baseline in Weekly Zolpidem Dosage During Weeks 5-6

    Baseline and Weeks 5-6

  • Change From Baseline in Weekly Zolpidem Dosage During Weeks 7-8

    Baseline and Weeks 7-8

  • Change From Baseline in Weekly Zolpidem Dosage During Weeks 9-10

    Baseline and Weeks 9-10

  • +8 more secondary outcomes

Study Arms (2)

Ramelteon 8 mg QD and current Zolpidem therapy

EXPERIMENTAL

Zolpidem therapy will be reduced by dose, frequency, or both for up to 10 weeks.

Drug: Ramelteon and zolpidem

Placebo QD and current Zolpidem therapy

PLACEBO COMPARATOR

Zolpidem therapy will be reduced by dose, frequency, or both for up to 10 weeks.

Drug: Placebo and zolpidem

Interventions

Ramelteon 8 mg, tablets, orally, once daily and current zolpidem therapy incrementally reduced by dose, frequency, or both for up to 10 weeks.

Also known as: Rozerem™, TAK-375, Ambien®
Ramelteon 8 mg QD and current Zolpidem therapy

Ramelteon placebo-matching tablets, orally, once daily and current zolpidem therapy incrementally reduced by dose, frequency, or both for up to 10 weeks.

Also known as: Ambien®
Placebo QD and current Zolpidem therapy

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Chronic insomnia and taking greater than or equal to 10 mg zolpidem at least 4 times per week.
  • Has been prescribed zolpidem for difficulty in initiating sleep.
  • Must report chronic use of zolpidem greater than or equal to10 mg therapy for a minimum of 3 months prior to entry into Period 1 of the study.
  • Must have taken zolpidem greater than or equal to 10 mg therapy for at least 4 of 7 days each week of the 4 weeks immediately prior to entry into the double blind phase, Period 2.
  • Expressed a willingness to discontinue zolpidem therapy.
  • Habitual bedtime is between 9:00 PM and 1:00 AM based on sleep history.
  • Negative test result for hepatitis B surface antigen and hepatitis C virus antibody.
  • Females of childbearing potential who are sexually active must agree to use adequate contraception, and can neither be pregnant nor lactating from Screening throughout the duration of the study.

You may not qualify if:

  • Known hypersensitivity to ramelteon, zolpidem, or melatonin.
  • Participated in any other investigational study and/or taken any investigational drug within 30 days prior to the first dose of run-in study medication.
  • Sleep schedule changes required by employment (eg, shift worker) within 3 months prior to the first night of run-in study medication.
  • History of fibromyalgia, history of seizures, sleep apnea, restless leg syndrome, periodic leg syndrome, chronic obstructive pulmonary disease, schizophrenia, bipolar disorder, mental retardation, or cognitive disorder.
  • History of drug addiction or drug abuse within the past 12 months.
  • History of alcohol abuse within the past 12 months, as defined in Diagnostic and Statistical Manual of Mental Disorders, 4th Edition revised and/or regularly consumes more than 2 alcoholic drinks per day.
  • Current significant hepatic, renal, endocrine, cardiovascular, gastrointestinal, pulmonary, hematological, or metabolic disease, unless currently controlled and stable with protocol-allowed medication, within 30 days prior to the first night of run-in study medication.
  • Body mass index of less than 18 or greater than 34 (weight /height2).
  • Any clinically important abnormal finding as documented by a medical history, physical examination, electrocardiogram, or clinical laboratory tests, as determined by the investigator.
  • Positive hepatitis panel.
  • Known history of human immunodeficiency virus.
  • Any additional conditions(s) that in the investigator's opinion would affect:
  • sleep/wake function
  • prohibit the subject from completing the study
  • indicate that continuation in the study would not be in the best interests of the subject.
  • +18 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (41)

Unknown Facility

Hot Springs, Arkansas, United States

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Anaheim, California, United States

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Fountain Valley, California, United States

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La Mesa, California, United States

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Los Angeles, California, United States

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Redlands, California, United States

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San Diego, California, United States

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San Francisco, California, United States

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Santa Monica, California, United States

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Denver, Colorado, United States

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Clearwater, Florida, United States

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Hollywood, Florida, United States

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Kissimmee, Florida, United States

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Naples, Florida, United States

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Pembroke Pines, Florida, United States

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Winter Park, Florida, United States

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Atlanta, Georgia, United States

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Austell, Georgia, United States

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Boise, Idaho, United States

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Louisville, Kentucky, United States

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Metairie, Louisiana, United States

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Chevy Chase, Maryland, United States

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St Louis, Missouri, United States

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Lincoln, Nebraska, United States

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New York, New York, United States

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West Seneca, New York, United States

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Raleigh, North Carolina, United States

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Wilmington, North Carolina, United States

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Cincinnati, Ohio, United States

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Toledo, Ohio, United States

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Portland, Oregon, United States

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Philadelphia, Pennsylvania, United States

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Greer, South Carolina, United States

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Fayetteville, Tennessee, United States

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Austin, Texas, United States

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Dallas, Texas, United States

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Fort Worth, Texas, United States

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Houston, Texas, United States

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San Angelo, Texas, United States

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San Antonio, Texas, United States

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Salt Lake City, Utah, United States

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Related Links

MeSH Terms

Conditions

Sleep Initiation and Maintenance Disorders

Interventions

ramelteonZolpidem

Condition Hierarchy (Ancestors)

Sleep Disorders, IntrinsicDyssomniasSleep Wake DisordersNervous System DiseasesMental Disorders

Intervention Hierarchy (Ancestors)

PyridinesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Results Point of Contact

Title
Sr. VP, Clinical Science
Organization
Takeda Global Research and Development Center, Inc.

Study Officials

  • Medical Director Clinical Science

    Takeda Global Research & Development Center

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 4
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

June 25, 2007

First Posted

June 27, 2007

Study Start

April 1, 2007

Primary Completion

March 1, 2008

Study Completion

May 1, 2008

Last Updated

July 20, 2010

Results First Posted

July 17, 2009

Record last verified: 2010-07

Locations