NCT00430248

Brief Summary

The purpose of this study is to compare the efficacy and safety of febuxostat, once Daily (QD), to allopurinol in subjects with hyperuricemia and gout.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
2,269

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started Feb 2007

Shorter than P25 for phase_3

Geographic Reach
1 country

258 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

January 25, 2007

Completed
7 days until next milestone

First Posted

Study publicly available on registry

February 1, 2007

Completed
Same day until next milestone

Study Start

First participant enrolled

February 1, 2007

Completed
1.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 1, 2008

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

March 1, 2008

Completed
1.4 years until next milestone

Results Posted

Study results publicly available

July 16, 2009

Completed
Last Updated

February 2, 2012

Status Verified

January 1, 2012

Enrollment Period

1.1 years

First QC Date

January 25, 2007

Results QC Date

March 12, 2009

Last Update Submit

January 31, 2012

Conditions

Keywords

tophihyperuricemiauric acidDrug Therapy

Outcome Measures

Primary Outcomes (1)

  • Percentage of Subjects Whose Serum Urate Level is <6.0 Milligrams Per Deciliter (mg/dL) at the Final Visit.

    The percentage of subjects whose serum urate level was \<6.0 mg/dL at the Final Visit was summarized. The Final Visit was the last visit at which a serum urate value was collected.

    Last Visit on treatment (up to 6 months)

Secondary Outcomes (16)

  • Percentage of Renal Impairment Subjects Whose Final Visit Serum Urate Level is <6.0 mg/dl

    Last Visit on treatment (up to 6 months)

  • Percentage of Subjects Whose Serum Urate Levels Are <6.0 mg/dL at Month 2 Visit.

    Month 2

  • Percentage of Subjects Whose Serum Urate Levels Are <6.0 mg/dL at Month 4 Visit.

    Month 4

  • Percentage of Subjects Whose Serum Urate Levels Are <6.0 mg/dL at Month 6 Visit.

    Month 6

  • Percentage of Subjects Whose Serum Urate Levels Are <5.0 mg/dL at Month 2 Visit.

    Month 2

  • +11 more secondary outcomes

Study Arms (3)

Febuxostat 40 mg QD

EXPERIMENTAL
Drug: Febuxostat

Febuxostat 80 mg QD

EXPERIMENTAL
Drug: Febuxostat

Allopurinol 200 mg or 300 mg QD

ACTIVE COMPARATOR

(dependent on renal function)

Drug: Allopurinol

Interventions

Febuxostat 40 mg, capsules, orally, once daily for up to 6 months.

Also known as: TMX-67, Tei-6720, Uloric
Febuxostat 40 mg QD

Allopurinol 200 mg or 300 mg, capsules, orally, once daily for up to 6 months. Dose is dependent on the subject's renal function. Subjects with normal renal function or mild renal impairment received 300 mg once daily; subjects with moderate renal impairment received 200 mg once daily.

Also known as: Zyloprim
Allopurinol 200 mg or 300 mg QD

Eligibility Criteria

Age18 Years - 85 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Has one or more of the American Rheumatism Association criteria for the diagnosis of gout.
  • Females of childbearing potential who are sexually active must agree to use adequate contraception, and can neither be pregnant nor lactating from Screening throughout the duration of the study.
  • Must have a serum urate level greater than or equal to 8.0 milligram per deciliter (mg/dL).

You may not qualify if:

  • Have a severe, unstable, or life threatening medical condition that would likely prevent them from completing this study.
  • Has a known body reaction to febuxostat, allopurinol, naproxen, any other non-steroidal anti-inflammatory drug (NSAID), aspirin, lansoprazole, colchicine, or any components in their formulation.
  • History of xanthinuria.
  • Alcohol consumption greater than 14/week.
  • History of significant concomitant illness.
  • Active liver or peptic ulcer disease.
  • Has rheumatoid arthritis requiring treatment.
  • Has estimated creatinine clearance less than 30 milliliter per minute (mL/min) calculated using the Cockcroft-Gault formula corrected for ideal body weight.
  • Requires therapy with any other urate-lowering drug other than the study drug; long-term use of NSAIDs and COX-2 inhibitors; salicylates; thiazide diuretics; losartan; azathioprine; mercaptopurine; theophylline; intravenous (IV) colchicine; cyclosporine; cyclophosphamide; pyrazinamide; sulfamethoxazole;trimethoprim.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (258)

Unknown Facility

Birmingham, Alabama, United States

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Hoover, Alabama, United States

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Hueytown, Alabama, United States

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Huntsville, Alabama, United States

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Mobile, Alabama, United States

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Montgomery, Alabama, United States

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Northport, Alabama, United States

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Ozark, Alabama, United States

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Tuscaloosa, Alabama, United States

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Chandler, Arizona, United States

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Gilbert, Arizona, United States

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Mesa, Arizona, United States

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Peoria, Arizona, United States

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Phoenix, Arizona, United States

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Scottsdale, Arizona, United States

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Sierra Vista, Arizona, United States

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Tucson, Arizona, United States

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Fort Smith, Arkansas, United States

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Jonesboro, Arkansas, United States

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Little Rock, Arkansas, United States

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Anaheim, California, United States

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Carmichael, California, United States

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Clovis, California, United States

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Concord, California, United States

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El Centro, California, United States

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Fair Oaks, California, United States

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Fullerton, California, United States

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Huntington Beach, California, United States

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Irvine, California, United States

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La Jolla, California, United States

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Laguna Hills, California, United States

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Los Angeles, California, United States

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Pasadena, California, United States

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Rancho Cucamonga, California, United States

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Riverside, California, United States

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Sacramento, California, United States

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San Diego, California, United States

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San Luis Obispo, California, United States

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Santa Barbara, California, United States

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Santa Maria, California, United States

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Torrance, California, United States

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Tustin, California, United States

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Vallejo, California, United States

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Vista, California, United States

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Walnut Creek, California, United States

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West Covina, California, United States

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Westlake Village, California, United States

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Whittier, California, United States

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Boulder, Colorado, United States

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Colorado Springs, Colorado, United States

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Denver, Colorado, United States

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Highlands Ranch, Colorado, United States

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Littleton, Colorado, United States

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Longmont, Colorado, United States

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Wheat Ridge, Colorado, United States

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Danbury, Connecticut, United States

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Trumbull, Connecticut, United States

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Washington D.C., District of Columbia, United States

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Aventura, Florida, United States

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Boynton Beach, Florida, United States

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Brandon, Florida, United States

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Daytona Beach, Florida, United States

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DeLand, Florida, United States

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Delray Beach, Florida, United States

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Fort Lauderdale, Florida, United States

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Fort Myers, Florida, United States

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Gainsville, Florida, United States

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Hallandale, Florida, United States

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Hialeah, Florida, United States

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Holly Hill, Florida, United States

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Jupiter, Florida, United States

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Kissimmee, Florida, United States

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Largo, Florida, United States

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Miami, Florida, United States

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Naples, Florida, United States

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New Port Richey, Florida, United States

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New Smyrna Beach, Florida, United States

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Opa-locka, Florida, United States

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Orlando, Florida, United States

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South Miami, Florida, United States

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St. Petersburg, Florida, United States

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Tallahassee, Florida, United States

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Tampa, Florida, United States

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West Palm Beach, Florida, United States

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Winter Haven, Florida, United States

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Zephyrhills, Florida, United States

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Atlanta, Georgia, United States

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Conyers, Georgia, United States

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Decatur, Georgia, United States

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Dunwoody, Georgia, United States

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Gainesville, Georgia, United States

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Marietta, Georgia, United States

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Stockbridge, Georgia, United States

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Honolulu, Hawaii, United States

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Boise, Idaho, United States

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Coeur d'Alene, Idaho, United States

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Meridian, Idaho, United States

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Nampa, Idaho, United States

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Arlington Heights, Illinois, United States

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Chicago, Illinois, United States

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Evanston, Illinois, United States

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Springfield, Illinois, United States

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Vernon Hills, Illinois, United States

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Elkhart, Indiana, United States

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Evansville, Indiana, United States

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Mishawaka, Indiana, United States

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Clive, Iowa, United States

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Des Moines, Iowa, United States

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Dubuque, Iowa, United States

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Kansas City, Kansas, United States

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Wichita, Kansas, United States

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Elizabethtown, Kentucky, United States

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Lexington, Kentucky, United States

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Louisville, Kentucky, United States

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Baton Rouge, Louisiana, United States

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Metairie, Louisiana, United States

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New Orleans, Louisiana, United States

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Ruston, Louisiana, United States

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Shreveport, Louisiana, United States

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Slidell, Louisiana, United States

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Baltimore, Maryland, United States

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Frederick, Maryland, United States

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Owings Mills, Maryland, United States

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Prince Frederick, Maryland, United States

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Wheaton, Maryland, United States

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Fall River, Massachusetts, United States

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New Bedford, Massachusetts, United States

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Springfield, Massachusetts, United States

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Worcester, Massachusetts, United States

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Ann Arbor, Michigan, United States

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Flint, Michigan, United States

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Kalamazoo, Michigan, United States

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Lansing, Michigan, United States

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Stevensville, Michigan, United States

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Troy, Michigan, United States

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Chaska, Minnesota, United States

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Flowood, Mississippi, United States

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Jackson, Mississippi, United States

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Olive Branch, Mississippi, United States

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Florissant, Missouri, United States

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Jefferson City, Missouri, United States

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Manchester, Missouri, United States

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Mexico, Missouri, United States

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St Louis, Missouri, United States

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Billings, Montana, United States

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Butte, Montana, United States

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Grand Island, Nebraska, United States

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Lincoln, Nebraska, United States

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Omaha, Nebraska, United States

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Las Vegas, Nevada, United States

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Reno, Nevada, United States

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Dover, New Hampshire, United States

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Blackwood, New Jersey, United States

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Edison, New Jersey, United States

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Flemington, New Jersey, United States

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Manalapan, New Jersey, United States

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Medford, New Jersey, United States

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Midland Park, New Jersey, United States

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Albuquerque, New Mexico, United States

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Endwell, New York, United States

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Mineola, New York, United States

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New York, New York, United States

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Smithtown, New York, United States

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Syracuse, New York, United States

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Charlotte, North Carolina, United States

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Greensboro, North Carolina, United States

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Greenville, North Carolina, United States

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Harrisburg, North Carolina, United States

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High Point, North Carolina, United States

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Lenoir, North Carolina, United States

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Raleigh, North Carolina, United States

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Winston-Salem, North Carolina, United States

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Austintown, Ohio, United States

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Beachwood, Ohio, United States

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Chardon, Ohio, United States

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Cincinnati, Ohio, United States

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Cleveland, Ohio, United States

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Dayton, Ohio, United States

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Hudson, Ohio, United States

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Kettering, Ohio, United States

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Lyndhurst, Ohio, United States

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Perrysburg, Ohio, United States

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Toledo, Ohio, United States

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Willoughby Hills, Ohio, United States

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Youngstown, Ohio, United States

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Oklahoma City, Oklahoma, United States

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Tulsa, Oklahoma, United States

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Bend, Oregon, United States

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Eugene, Oregon, United States

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Lake Oswego, Oregon, United States

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Medford, Oregon, United States

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Portland, Oregon, United States

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Bethlehem, Pennsylvania, United States

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Duncansville, Pennsylvania, United States

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East Norriton, Pennsylvania, United States

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Feasterville-Trevose, Pennsylvania, United States

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Harrisburg, Pennsylvania, United States

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Lansdale, Pennsylvania, United States

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Mechanicsburg, Pennsylvania, United States

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Morrisville, Pennsylvania, United States

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Penndel, Pennsylvania, United States

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Philadelphia, Pennsylvania, United States

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Pittsburgh, Pennsylvania, United States

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Reading, Pennsylvania, United States

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Scotland, Pennsylvania, United States

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West Reading, Pennsylvania, United States

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Cranston, Rhode Island, United States

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East Providence, Rhode Island, United States

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Charleston, South Carolina, United States

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Columbia, South Carolina, United States

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Greenville, South Carolina, United States

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Greer, South Carolina, United States

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Mt. Pleasant, South Carolina, United States

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Orangeburg, South Carolina, United States

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Simpsonville, South Carolina, United States

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Spartanburg, South Carolina, United States

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Bristol, Tennessee, United States

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Chattanooga, Tennessee, United States

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Clarksville, Tennessee, United States

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Collierville, Tennessee, United States

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Jackson, Tennessee, United States

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Johnson City, Tennessee, United States

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Memphis, Tennessee, United States

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Nashville, Tennessee, United States

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New Tazewell, Tennessee, United States

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Amarillo, Texas, United States

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Austin, Texas, United States

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Beaumont, Texas, United States

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Bellaire, Texas, United States

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Bryan, Texas, United States

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Dallas, Texas, United States

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El Paso, Texas, United States

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Fort Worth, Texas, United States

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Houston, Texas, United States

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Killeen, Texas, United States

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Lake Jackson, Texas, United States

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Odessa, Texas, United States

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San Antonio, Texas, United States

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Sugar Land, Texas, United States

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Waco, Texas, United States

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Layton, Utah, United States

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Midvale, Utah, United States

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Salt Lake City, Utah, United States

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St. George, Utah, United States

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West Jordan, Utah, United States

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Chesapeake, Virginia, United States

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Newport News, Virginia, United States

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Norfolk, Virginia, United States

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Richmond, Virginia, United States

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Everett, Washington, United States

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Gig Harbor, Washington, United States

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Lakewood, Washington, United States

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Olympia, Washington, United States

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Spokane, Washington, United States

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Tacoma, Washington, United States

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Vancouver, Washington, United States

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Monroe, Wisconsin, United States

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Oregon, Wisconsin, United States

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Related Publications (7)

  • Becker MA, Schumacher HR, Espinoza LR, Wells AF, MacDonald P, Lloyd E, Lademacher C. The urate-lowering efficacy and safety of febuxostat in the treatment of the hyperuricemia of gout: the CONFIRMS trial. Arthritis Res Ther. 2010;12(2):R63. doi: 10.1186/ar2978. Epub 2010 Apr 6.

  • Wortmann RL, Macdonald PA, Hunt B, Jackson RL. Effect of prophylaxis on gout flares after the initiation of urate-lowering therapy: analysis of data from three phase III trials. Clin Ther. 2010 Dec;32(14):2386-97. doi: 10.1016/j.clinthera.2011.01.008.

  • Becker MA, MacDonald PA, Hunt B, Gunawardhana L. Treating hyperuricemia of gout: safety and efficacy of febuxostat and allopurinol in older versus younger subjects. Nucleosides Nucleotides Nucleic Acids. 2011 Dec;30(12):1011-7. doi: 10.1080/15257770.2011.603715.

  • Chohan S, Becker MA, MacDonald PA, Chefo S, Jackson RL. Women with gout: efficacy and safety of urate-lowering with febuxostat and allopurinol. Arthritis Care Res (Hoboken). 2012 Feb;64(2):256-61. doi: 10.1002/acr.20680.

  • Becker MA, MacDonald PA, Hunt BJ, Jackson RL. Diabetes and gout: efficacy and safety of febuxostat and allopurinol. Diabetes Obes Metab. 2013 Nov;15(11):1049-55. doi: 10.1111/dom.12135. Epub 2013 Jun 12.

  • Jackson RL, Hunt B, MacDonald PA. The efficacy and safety of febuxostat for urate lowering in gout patients >/=65 years of age. BMC Geriatr. 2012 Mar 21;12:11. doi: 10.1186/1471-2318-12-11.

  • Wells AF, MacDonald PA, Chefo S, Jackson RL. African American patients with gout: efficacy and safety of febuxostat vs allopurinol. BMC Musculoskelet Disord. 2012 Feb 9;13:15. doi: 10.1186/1471-2474-13-15.

Related Links

MeSH Terms

Conditions

GoutHyperuricemia

Interventions

FebuxostatAllopurinol

Condition Hierarchy (Ancestors)

ArthritisJoint DiseasesMusculoskeletal DiseasesCrystal ArthropathiesRheumatic DiseasesPurine-Pyrimidine Metabolism, Inborn ErrorsMetabolism, Inborn ErrorsGenetic Diseases, InbornCongenital, Hereditary, and Neonatal Diseases and AbnormalitiesMetabolic DiseasesNutritional and Metabolic DiseasesPathologic ProcessesPathological Conditions, Signs and Symptoms

Intervention Hierarchy (Ancestors)

ThiazolesSulfur CompoundsOrganic ChemicalsAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPurinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-Ring

Results Point of Contact

Title
Sr. VP, Clinical Sciences
Organization
Takeda Global Research and Development Center, Inc.

Study Officials

  • Medical Director

    Takeda

    STUDY CHAIR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 25, 2007

First Posted

February 1, 2007

Study Start

February 1, 2007

Primary Completion

March 1, 2008

Study Completion

March 1, 2008

Last Updated

February 2, 2012

Results First Posted

July 16, 2009

Record last verified: 2012-01

Locations