NCT00347360

Brief Summary

This is a randomized, double-blind, double-dummy, parallel group trial employing 15 cells of a 4x4 factorial design (no placebo)to compare the hypertensive effects in patients with Stage 1 and Stage 2 hypertension of carvedilol (20, 40 or 80 mg daily) alone, lisinopril (10, 20 or 40 mg daily) alone, and all combinations of the doses.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
654

participants targeted

Target at P75+ for phase_3 hypertension

Timeline
Completed

Started Jul 2006

Typical duration for phase_3 hypertension

Geographic Reach
1 country

151 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

June 29, 2006

Completed
2 days until next milestone

Study Start

First participant enrolled

July 1, 2006

Completed
3 days until next milestone

First Posted

Study publicly available on registry

July 4, 2006

Completed
1.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 1, 2008

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

April 1, 2008

Completed
1.6 years until next milestone

Results Posted

Study results publicly available

November 9, 2009

Completed
Last Updated

December 26, 2016

Status Verified

November 1, 2016

Enrollment Period

1.8 years

First QC Date

June 29, 2006

Results QC Date

April 22, 2009

Last Update Submit

November 3, 2016

Conditions

Keywords

carvedilolhypertensionlisinoprilfactorial

Outcome Measures

Primary Outcomes (2)

  • Change From Baseline to Week 6 in 24 Hour (hr) Mean Diastolic Blood Pressure

    Ambulatory blood pressure monitoring (ABPM) was completed at Baseline and at the end of treatment/Week 6 or early withdrawal by standard electronic ABPM equipment worn by the subject for 24-hr of ambulatory activity. The 24 hr assessment period started at the time of the first reading and ended exactly 24 hr later on the following day. Data collected included mean diastolic blood pressure (DBP).

    Baseline, Week 6.

  • Change From Baseline to Week 6 in Trough Diastolic Blood Pressure

    Trough ABPM was the average across 20-24 hr after dosing for each subject.

    Baseline, Week 6

Secondary Outcomes (10)

  • Change From Baseline to Week 6 in 24 Hour Mean Systolic Blood Pressure

    Baseline, Week 6

  • Change From Baseline to Week 6 in Trough Systolic Blood Pressure

    Baseline, Week 6

  • Dose-response Treatment Estimates: Change From Baseline to Week 6 in 24 Hour Mean DBP by ABPM (Ambulatory Blood Pressure Monitoring)

    Baseline, Week 6

  • Change From Baseline to Week 6 in Trough to Peak Ratios of DBP by 24 Hour ABPM (Ambulatory Blood Pressure Monitoring)

    Baseline, Week 6

  • Overall Description of Safety in Each Treatment Group Using Adverse Events, Laboratory Evaluations, ECG Changes, Vital Sign Changes, and Withdrawal Rates.

    Weeks 1 through 48

  • +5 more secondary outcomes

Study Arms (2)

lisinopril

EXPERIMENTAL

lisinopril

Drug: lisinopril

carvedilol

EXPERIMENTAL

carvedilol controlled release formulation

Drug: carvedilol controlled release formulation

Interventions

lisinopril
Also known as: lisinopril
carvedilol

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Subject has given signed informed consent.
  • Subject is male or female 18 years of age at the time informed consent is signed.
  • At the Screening visit, subject has a documented history or current presentation with stage 1 or stage 2 hypertension (see Section 15.1, Appendix 1 and Section 15.4, Appendix 4) which meets one of the following criteria. Note: All blood pressures are mean sitting cuff pressures:
  • Documented history of hypertension and receiving two antihypertensive medications with mean sDBP \<90 mmHg or for diabetic subjects (defined as having an established diagnosis of diabetes or receiving treatment for diabetes), mean sDBP \<80 mmHg. Subjects taking beta blockers, clonidine, or other antihypertensive medications where abrupt discontinuation would be of clinical concern must be tapered off the medication during the Washout/Placebo Run-in phase to avoid rebound hypertension. All subjects must be able to be safely withdrawn from all antihypertensive treatment during the Washout/Placebo Run-in phase. Subjects should not be enrolled if the investigator thinks it is likely the subject's mean sDBP will exceed 109 mmHg or their mean sSBP will exceed 180 mmHg during the Washout/Placebo Run-in phase (NOTE: A combination drug containing two antihypertensive agents represents two antihypertensive medications \[e.g., Hyzaar is losartan potassium AND hydrochlorothiazide, therefore, counts as two antihypertensive medications\].) OR Receiving one antihypertensive medication with mean sDBP =109 mmHg and can be safely withdrawn from all antihypertensive medication during the Washout/Placebo Run-in phase. Any subject who is receiving beta-blockers, clonidine, or other antihypertensive medications where abrupt discontinuation would be of clinical concern must have the dose tapered down during the Washout/Placebo Run-in phase to avoid rebound hypertension. All subjects must be able to be safely withdrawn from all antihypertensive treatment during the Washout/Placebo Run-in phase. Subjects should not be enrolled if the investigator thinks it is likely the subject's mean sDBP will exceed 109 mmHg or their mean sSBP will exceed 180 mmHg during the Washout/Placebo Run-in phase.
  • (NOTE: A combination drug containing two antihypertensive agents represents two antihypertensive medications \[e.g., Hyzaar is losartan potassium AND hydrochlorothiazide, therefore, counts as two antihypertensive medications\].
  • OR Untreated/newly diagnosed subjects: mean sDBP =95 and =109, or for diabetic subjects, mean sDBP =85 and =109 (see Section 15.1, Appendix 1). If newly diagnosed, must have qualifying blood pressure confirmed on two consecutive visits with the mean sDBP value not differing more than 8 mmHg. (Previously untreated subjects include subjects who have not been treated for hypertension in the last two months.).
  • At Baseline:
  • AND
  • RANDOMIZATON DAY: After completion of the ABPM assessment, subject meets the following ABPM (both 12 hr and 24 hr) criteria (see Section 15.1, Appendix 1):
  • Mean 12-hour daytime (9 AM to 9 PM) DBP ≥90 and ≤109mmHg (or for diabetic subjects, ≥80 and ≤109mmHg)
  • At least 75% of the programmed readings properly recorded over 24-hour monitoring period
  • No more than two non-consecutive hours with less than two successful readings per hour while awake, and no more than two consecutive hours with less than one successful reading per hour during the sleep period over the 24-hour monitoring period
  • At least two successful readings per hour for three of the last four hours of recording (trough period i.e., 20-24 hour during which subjects must be awake) with a total of at least 7 successful readings over this period.

You may not qualify if:

  • Subject is taking ≥3 antihypertensive medications. (NOTE: A combination drug containing two antihypertensive agents represents two antihypertensive medications \[e.g., Hyzaar is losartan potassium AND hydrochlorothiazide, therefore, counts as two antihypertensive medications\].)
  • Subject has DBP =90 mmHg (or for diabetic subjects, DBP =80 mmHg) on two antihypertensive medications.
  • Subject has any known contraindication to ACE inhibitors (e.g., ACE-induced cough, angioedema or negative renal effects), or blocker treatment.
  • Hyperkalemia or history of hyperkalemia resulting from either Type IV RTA (renal tubular acidosis) or previous ACEi therapy.
  • Is female of childbearing potential. NOTE: Female subjects who are postmenopausal (i.e., no menstrual period for a minimum of 12 months prior to Screening) or surgically sterilized are eligible for the study. If judged appropriate, a postmenopausal woman may be required to have a documented negative urine pregnancy test.
  • Subject has malignant (accelerated) hypertension, history of malignant hypertension, or secondary forms of hypertension.
  • Subject has mean sitting SBP =180 mmHg.
  • Subject has advanced hypertensive retinopathy (Keith Wagner Grade IV).
  • Subject has Type 1 diabetes mellitus, or those with Type 2 having HbA1c ≥9% at Screening.
  • Subject has uncorrected primary obstructive or severe regurgitative valvular disease, nondilated (restrictive) or hypertrophic cardiomyopathies.
  • Subject has any of the following conditions:
  • uncontrollable or symptomatic arrhythmias unstable angina or angina treated with a beta-blocker sick sinus syndrome or second or third degree heart block (unless treated with a permanent, functioning pacemaker) bradycardia (sitting heart rate \<55 bpm) history of myocardial infarction stroke within 3 months of Screening
  • Subject is in atrial fibrillation.
  • Subject has Congestive Heart Failure NYHA (New York Heart Association) class II-IV \[The Criteria Committee of the New York Heart Association, 1994\].
  • Current clinical evidence of asthma or chronic obstructive pulmonary disease (e.g., severe emphysema or chronic bronchitis) requiring long term use of inhaled oral bronchodilator or steroid drug therapy; also subjects with a history of bronchospastic disease not undergoing active therapy in whom, in the investigator's opinion, treatment with the study medication could provoke bronchospasm; or requirement for or anticipated treatment with beta-2 agonist therapy (e.g., albuterol \[Ventolin, Proventil\], metaproterenol \[Alupent\], pirbuterol \[Maxair\], terbutaline \[Brethaire\], isoetharine \[Bronkosol\], and Levalbuterol \[Xopenex\]).
  • +9 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (151)

GSK Investigational Site

Anniston, Alabama, 36207, United States

Location

GSK Investigational Site

Birmingham, Alabama, 35215, United States

Location

GSK Investigational Site

Birmingham, Alabama, 35216, United States

Location

GSK Investigational Site

Birmingham, Alabama, 35235, United States

Location

GSK Investigational Site

Birmingham, Alabama, 35242, United States

Location

GSK Investigational Site

Haleyville, Alabama, 35565, United States

Location

GSK Investigational Site

Mobile, Alabama, 36617, United States

Location

GSK Investigational Site

Muscle Shoals, Alabama, 35662, United States

Location

GSK Investigational Site

Chandler, Arizona, 85225, United States

Location

GSK Investigational Site

Gilbert, Arizona, 85296, United States

Location

GSK Investigational Site

Glendale, Arizona, 85308, United States

Location

GSK Investigational Site

Mesa, Arizona, 85206, United States

Location

GSK Investigational Site

Phoenix, Arizona, 85023, United States

Location

GSK Investigational Site

Phoenix, Arizona, 85032, United States

Location

GSK Investigational Site

Phoenix, Arizona, Arizona, 86106, United States

Location

GSK Investigational Site

Scottsdale, Arizona, 85251, United States

Location

GSK Investigational Site

Scottsdale, Arizona, 85260, United States

Location

GSK Investigational Site

Sun City, Arizona, 85351, United States

Location

GSK Investigational Site

Tucson, Arizona, 85712, United States

Location

GSK Investigational Site

Tucson, Arizona, 85741, United States

Location

GSK Investigational Site

Little Rock, Arkansas, 72204, United States

Location

GSK Investigational Site

Searcy, Arkansas, 72143, United States

Location

GSK Investigational Site

Beuna Park, California, 90620, United States

Location

GSK Investigational Site

Beverly Hills, California, 90211, United States

Location

GSK Investigational Site

Burbank, California, 91505, United States

Location

GSK Investigational Site

Carlsbad, California, 92008, United States

Location

GSK Investigational Site

Fountain Valley, California, 92708, United States

Location

GSK Investigational Site

Fresno, California, 93703, United States

Location

GSK Investigational Site

Loma Linda, California, 92354, United States

Location

GSK Investigational Site

Mission Viejo, California, 92691, United States

Location

GSK Investigational Site

Pico Rivera, California, 90660, United States

Location

GSK Investigational Site

Rancho Cordova, California, 95670, United States

Location

GSK Investigational Site

San Diego, California, 92117, United States

Location

GSK Investigational Site

San Diego, California, 92128, United States

Location

GSK Investigational Site

Santa Ana, California, 92705, United States

Location

GSK Investigational Site

Vista, California, 92084, United States

Location

GSK Investigational Site

Walnut Creek, California, 94598, United States

Location

GSK Investigational Site

Colorado Springs, Colorado, 80904, United States

Location

GSK Investigational Site

Denver, Colorado, 80206, United States

Location

GSK Investigational Site

Wilmington, Delaware, 19805, United States

Location

GSK Investigational Site

Washington D.C., District of Columbia, 20017, United States

Location

GSK Investigational Site

Coral Gables, Florida, 33134, United States

Location

GSK Investigational Site

Hialeah, Florida, 33013, United States

Location

GSK Investigational Site

Hollywood, Florida, 33023, United States

Location

GSK Investigational Site

Jacksonville, Florida, 32205, United States

Location

GSK Investigational Site

Jacksonville Beach, Florida, 32250, United States

Location

GSK Investigational Site

Miami, Florida, 33156, United States

Location

GSK Investigational Site

Miami, Florida, 33169, United States

Location

GSK Investigational Site

Palm Harbor, Florida, 34684, United States

Location

GSK Investigational Site

Pembroke Pines, Florida, 33024, United States

Location

GSK Investigational Site

Pembroke Pines, Florida, 33027, United States

Location

GSK Investigational Site

Sarasota, Florida, 34239, United States

Location

GSK Investigational Site

West Palm Beach, Florida, 33409, United States

Location

GSK Investigational Site

Gainesville, Georgia, 30501, United States

Location

GSK Investigational Site

Marietta, Georgia, 30066, United States

Location

GSK Investigational Site

Sandersville, Georgia, 31082, United States

Location

GSK Investigational Site

Savannah, Georgia, 31406, United States

Location

GSK Investigational Site

Aurora, Illinois, 60504, United States

Location

GSK Investigational Site

Chicago, Illinois, 60607, United States

Location

GSK Investigational Site

Chicago, Illinois, 60610, United States

Location

GSK Investigational Site

Melrose Park, Illinois, 60160, United States

Location

GSK Investigational Site

Avon, Indiana, 46123, United States

Location

GSK Investigational Site

Bloomington, Indiana, 47102, United States

Location

GSK Investigational Site

Fort Wayne, Indiana, 46804, United States

Location

GSK Investigational Site

Indianapolis, Indiana, 46250, United States

Location

GSK Investigational Site

Ames, Iowa, 50010, United States

Location

GSK Investigational Site

Wichita, Kansas, 67205, United States

Location

GSK Investigational Site

Slidell, Louisiana, 70458, United States

Location

GSK Investigational Site

Springfield, Massachusetts, 01103, United States

Location

GSK Investigational Site

Taunton, Massachusetts, 02780., United States

Location

GSK Investigational Site

Bingham Farms, Michigan, 48025, United States

Location

GSK Investigational Site

Brooklyn Center, Minnesota, 55430, United States

Location

GSK Investigational Site

Missoula, Montana, 59808, United States

Location

GSK Investigational Site

O Fallon, Montana, 63366, United States

Location

GSK Investigational Site

Omaha, Nebraska, 68131, United States

Location

GSK Investigational Site

Las Vegas, Nevada, 89016, United States

Location

GSK Investigational Site

Las Vegas, Nevada, 89119, United States

Location

GSK Investigational Site

Las Vegas, Nevada, 89128, United States

Location

GSK Investigational Site

Cherry Hill, New Jersey, 08034, United States

Location

GSK Investigational Site

Edison, New Jersey, 08817, United States

Location

GSK Investigational Site

Ridgewood, New Jersey, 7450, United States

Location

GSK Investigational Site

Voorhees Township, New Jersey, 08043, United States

Location

GSK Investigational Site

Albuquerque, New Mexico, 87102, United States

Location

GSK Investigational Site

Brooklyn, New York, 11203, United States

Location

GSK Investigational Site

Buffalo, New York, 14215, United States

Location

GSK Investigational Site

Kingston, New York, 12401, United States

Location

GSK Investigational Site

Lewinston, New York, 14092, United States

Location

GSK Investigational Site

Tonawanda, New York, 14150-1810, United States

Location

GSK Investigational Site

Asheville, North Carolina, 28801, United States

Location

GSK Investigational Site

Charlotte, North Carolina, 28211, United States

Location

GSK Investigational Site

High Point, North Carolina, 27262, United States

Location

GSK Investigational Site

Raleigh, North Carolina, 27615, United States

Location

GSK Investigational Site

Fargo, North Dakota, 58103, United States

Location

GSK Investigational Site

Cincinnati, Ohio, 45219, United States

Location

GSK Investigational Site

Cincinnati, Ohio, 45236, United States

Location

GSK Investigational Site

Cleveland, Ohio, 44106, United States

Location

GSK Investigational Site

Cleveland, Ohio, 44195, United States

Location

GSK Investigational Site

Dayton, Ohio, 45406, United States

Location

GSK Investigational Site

Oklahoma City, Oklahoma, 73103, United States

Location

GSK Investigational Site

Oklahoma City, Oklahoma, 73112, United States

Location

GSK Investigational Site

Tulsa, Oklahoma, 74104, United States

Location

GSK Investigational Site

Eugene, Oregon, 97401, United States

Location

GSK Investigational Site

Beaver, Pennsylvania, 15009, United States

Location

GSK Investigational Site

Doylestown, Pennsylvania, 18901, United States

Location

GSK Investigational Site

Erie, Pennsylvania, 16504, United States

Location

GSK Investigational Site

Havertown, Pennsylvania, 19083, United States

Location

GSK Investigational Site

Landsdale, Pennsylvania, 19446, United States

Location

GSK Investigational Site

Leetsdale, Pennsylvania, 15056, United States

Location

GSK Investigational Site

Philadelphia, Pennsylvania, 19152, United States

Location

GSK Investigational Site

Philadelphia, Pennsylvania, 19154, United States

Location

GSK Investigational Site

Warminster, Pennsylvania, 18974, United States

Location

GSK Investigational Site

West Chester, Pennsylvania, 19380, United States

Location

GSK Investigational Site

Beaufort, South Carolina, 29906, United States

Location

GSK Investigational Site

Charleston, South Carolina, 29403, United States

Location

GSK Investigational Site

Columbia, South Carolina, 29201, United States

Location

GSK Investigational Site

Gaffney, South Carolina, 29340, United States

Location

GSK Investigational Site

Greer, South Carolina, 29651, United States

Location

GSK Investigational Site

Hilton Head Island, South Carolina, 29926, United States

Location

GSK Investigational Site

Manning, South Carolina, 29102, United States

Location

GSK Investigational Site

Simpsonville, South Carolina, 29681, United States

Location

GSK Investigational Site

Spartanburg, South Carolina, 29303, United States

Location

GSK Investigational Site

Sumter, South Carolina, 29150, United States

Location

GSK Investigational Site

Taylors, South Carolina, 29687, United States

Location

GSK Investigational Site

Union, South Carolina, 29309, United States

Location

GSK Investigational Site

Clarksville, Tennessee, 37043, United States

Location

GSK Investigational Site

Jackson, Tennessee, 38305, United States

Location

GSK Investigational Site

Johnson City, Tennessee, 37601, United States

Location

GSK Investigational Site

Nashville, Tennessee, 37203, United States

Location

GSK Investigational Site

Selmer, Tennessee, 38375, United States

Location

GSK Investigational Site

Arlington, Texas, 76014, United States

Location

GSK Investigational Site

Austin, Texas, 78705, United States

Location

GSK Investigational Site

Georgetown, Texas, 78626, United States

Location

GSK Investigational Site

Grand Prairie/Texas, Texas, 5052, United States

Location

GSK Investigational Site

Houston, Texas, 77081, United States

Location

GSK Investigational Site

Longview, Texas, 75605, United States

Location

GSK Investigational Site

San Antonio, Texas, 78224, United States

Location

GSK Investigational Site

San Antonio, Texas, 78229, United States

Location

GSK Investigational Site

Sugar Land, Texas, 77479, United States

Location

GSK Investigational Site

Temple, Texas, 76502, United States

Location

GSK Investigational Site

Waco, Texas, 76712, United States

Location

GSK Investigational Site

Murray, Utah, 84107, United States

Location

GSK Investigational Site

Salt Lake City, Utah, 84102, United States

Location

GSK Investigational Site

Sandy City, Utah, 84094, United States

Location

GSK Investigational Site

Arlington, Virginia, 22205, United States

Location

GSK Investigational Site

Burke, Virginia, 22015, United States

Location

GSK Investigational Site

Chester, Virginia, 23836, United States

Location

GSK Investigational Site

Fairfax, Virginia, 22030, United States

Location

GSK Investigational Site

Manassas, Virginia, 20110, United States

Location

GSK Investigational Site

Spokane, Washington, 99206, United States

Location

GSK Investigational Site

Tacoma, Washington, 98405, United States

Location

GSK Investigational Site

Milwaukee, Wisconsin, 53209, United States

Location

Related Publications (1)

  • Bakris GL, Iyengar M, Lukas MA, Ordronneau P, Weber MA. Effect of combining extended-release carvedilol and lisinopril in hypertension: results of the COSMOS study. J Clin Hypertens (Greenwich). 2010 Sep;12(9):678-86. doi: 10.1111/j.1751-7176.2010.00341.x. Epub 2010 Jul 8.

Related Links

MeSH Terms

Conditions

Hypertension

Interventions

Lisinopril

Condition Hierarchy (Ancestors)

Vascular DiseasesCardiovascular Diseases

Intervention Hierarchy (Ancestors)

DipeptidesOligopeptidesPeptidesAmino Acids, Peptides, and Proteins

Results Point of Contact

Title
GSK Response Center
Organization
GlaxoSmithKline

Study Officials

  • GSK Clinical Trials

    GlaxoSmithKline

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 29, 2006

First Posted

July 4, 2006

Study Start

July 1, 2006

Primary Completion

April 1, 2008

Study Completion

April 1, 2008

Last Updated

December 26, 2016

Results First Posted

November 9, 2009

Record last verified: 2016-11

Data Sharing

IPD Sharing
Will share

Patient-level data for this study will be made available through www.clinicalstudydatarequest.com following the timelines and process described on this site.

Available IPD Datasets

Informed Consent Form (CFD105453)Access
Annotated Case Report Form (CFD105453)Access
Statistical Analysis Plan (CFD105453)Access
Individual Participant Data Set (CFD105453)Access
Study Protocol (CFD105453)Access
Clinical Study Report (CFD105453)Access
Dataset Specification (CFD105453)Access

Locations