NCT00093197

Brief Summary

Restoring blood flow to coronary arteries as quickly as possible is the best way to reduce the damage to the muscle that occurs with a heart attack. However, up to 25-50% of patients who have angioplasty may have ongoing damage to the heart muscle when the blockage is opened and blood flow is restored. Complications which may result from this ongoing damage include a larger area of damaged muscle in the heart, enlargement of the heart, an increased risk of death, and an increased risk of heart failure. Some of the ongoing damage may involve increased levels of the protein kinase C (PKC) enzyme. KAI-9803 is a selective inhibitor of delta PKC. In this study, delta PKC is used with angioplasty and other standard procedures to restore blood flow after a heart attack. This study is designed to evaluate safety of different amounts of KAI-9803 when used in treating heart attack patients undergoing angioplasty. We will also try to evaluate whether KAI-9803 can reduce the amount of heart muscle damage and the complications that may occur in these patients.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
154

participants targeted

Target at P75+ for phase_1

Timeline
Completed

Started Sep 2004

Typical duration for phase_1

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

September 1, 2004

Completed
1 month until next milestone

First Submitted

Initial submission to the registry

October 4, 2004

Completed
3 days until next milestone

First Posted

Study publicly available on registry

October 7, 2004

Completed
2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 1, 2006

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

October 1, 2006

Completed
Last Updated

September 2, 2011

Status Verified

August 1, 2011

Enrollment Period

2.1 years

First QC Date

October 4, 2004

Last Update Submit

August 31, 2011

Conditions

Outcome Measures

Primary Outcomes (2)

  • Number of participants with adverse events

    30 days

  • Number of participants with major cardiac events (death, congestive heart failure, recurrent myocardial infarction, repeat target vessel revascularization)

    6 months

Secondary Outcomes (5)

  • Creatine kinase-myocardial band (CK-MB)

    7 days or hospitalization discharge, whichever occurs first

  • ST-segment elevation

    24 hours

  • Angiography vessel flow

    Day 1

  • Infarct size by single photon emission computed tomography (SPECT)

    14 days

  • Echocardiographic left ventricular ejection fraction (LVEF)

    14 days

Study Arms (5)

A1: KAI-9803

EXPERIMENTAL
Drug: KAI-9803 for Injection

A2: KAI-9803

EXPERIMENTAL
Drug: KAI-9803 for Injection

A3: KAI-9803

EXPERIMENTAL
Drug: KAI-9803 for Injection

A4: KAI-9803

EXPERIMENTAL
Drug: KAI-9803 for Injection

A5: Placebo

PLACEBO COMPARATOR
Drug: Placebo

Interventions

0.05 mg

A1: KAI-9803
A5: Placebo

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Symptoms of cardiac ischemia at rest or with increasing frequency (angina or angina equivalent), with episodes lasting for at least 30 minutes within 6 hours of presentation
  • Persistent ST-segment elevation of ≥ 0.2 mV in at least 2 contiguous precordial leads indicative of anterior Myocardial Infarction (MI) location (leads V1-V4)
  • At least 18 years old
  • Complete occlusion of the left anterior descending artery (Thrombolysis in Myocardial Infarction (TIMI) 0-1 flow) demonstrated on the initial angiogram
  • Culprit lesion suitable for primary percutaneous coronary intervention (PCI)

You may not qualify if:

  • Any left bundle branch block (new or old), intraventricular conduction defect, or paced rhythm that would obscure the diagnosis of acute anterior ST Elevation Myocardial Infarction (STEMI)
  • Any prior documented myocardial infarction (MI), including old Q waves documented on prior ECGs or a clinical history of definite MI
  • Any prior coronary artery bypass grafting (CABG)
  • Cardiogenic shock at initial hospital presentation, consisting of persistent hypotension (systolic blood pressure \< 90 mm Hg for \> 20 minutes) and signs of end-organ dysfunction (oliguria, altered mental status, poor peripheral perfusion, and lactic acidosis)
  • TIMI grade 2 or 3 flow in the left anterior descending artery documented on the initial diagnostic angiogram
  • Culprit lesion in the left anterior descending artery that is not suitable for primary PCI
  • Treatment with intravenous fibrinolytic therapy (i.e. alteplase, reteplase, tenecteplase, or streptokinase) within the 24 hours before presentation
  • Pregnancy
  • Know baseline creatinine \> 2.5 mg/dL without renal dialysis/renal replacement therapy within the 30 days before presentation
  • Inability to comply with study procedures, inability to undergo cardiac catheterization or primary percutaneous coronary intervention (PCI)
  • Participation in a study of experimental therapy (drug or device) within 30 days of presentation, or prior participation in this study

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Duke Clinical Research Institute

Durham, North Carolina, 27715, United States

Location

MeSH Terms

Conditions

Myocardial Infarction

Interventions

KAI 9803Injections

Condition Hierarchy (Ancestors)

Myocardial IschemiaHeart DiseasesCardiovascular DiseasesVascular DiseasesInfarctionIschemiaPathologic ProcessesPathological Conditions, Signs and SymptomsNecrosis

Intervention Hierarchy (Ancestors)

Drug Administration RoutesDrug TherapyTherapeutics

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 4, 2004

First Posted

October 7, 2004

Study Start

September 1, 2004

Primary Completion

October 1, 2006

Study Completion

October 1, 2006

Last Updated

September 2, 2011

Record last verified: 2011-08

Locations